Tetrazoles via Multicomponent Reactions

por Neochoritis, Constantinos G., Zhao, Ting, Dömling, Alexander
Publicado 2019

Atorvastatin (Lipitor) by MCR

por Zarganes-Tzitzikas, Tryfon, Neochoritis, Constantinos G., Dömling, Alexander
Publicado 2019

Multicomponent Reactions: “Kinderleicht”

por Neochoritis, Constantinos G., Zarganes-Tzitzikas, Tryfon, Katsampoxaki-Hodgetts, Kallia, Dömling, Alexander
Publicado 2020

Application of Silver Nanoparticles in the Multicomponent Reaction Domain: A Combined Catalytic Reduction Methodology to Efficiently Access Potential Hypertension or Inflammation I...

por Iordanidou, Domna, Zarganes-Tzitzikas, Tryfon, Neochoritis, Constantinos G., Dömling, Alexander, Lykakis, Ioannis N.
Publicado 2018

A multicomponent tetrazolo indole synthesis

por Lei, Xiaofang, Lampiri, Panagiota, Patil, Pravin, Angeli, Giasemi, Neochoritis, Constantinos G., Dömling, Alexander
Publicado 2021

Artificial Macrocycles as Potent p53–MDM2 Inhibitors

por Estrada-Ortiz, Natalia, Neochoritis, Constantinos G., Twarda-Clapa, Aleksandra, Musielak, Bogdan, Holak, Tad A., Dömling, Alexander
Publicado 2017

Multicomponent reaction–derived covalent inhibitor space

por Sutanto, Fandi, Shaabani, Shabnam, Neochoritis, Constantinos G., Zarganes-Tzitzikas, Tryfon, Patil, Pravin, Ghonchepour, Ehsan, Dömling, Alexander
Publicado 2021

Design of indole- and MCR-based macrocycles as p53-MDM2 antagonists

por Neochoritis, Constantinos G, Kazemi Miraki, Maryam, Abdelraheem, Eman M M, Surmiak, Ewa, Zarganes-Tzitzikas, Tryfon, Łabuzek, Beata, Holak, Tad A, Dömling, Alexander
Publicado 2019

Potential binding modes of the gut bacterial metabolite, 5-hydroxyindole, to the intestinal L-type calcium channels and its impact on the microbiota in rats

por Waclawiková, Barbora, Cesar Telles de Souza, Paulo, Schwalbe, Markus, Neochoritis, Constantinos G., Hoornenborg, Warner, Nelemans, Sieger A., Marrink, Siewert J., El Aidy, Sahar
Publicado 2022

Supported Gold Nanoparticle-Catalyzed Selective Reduction of Multifunctional, Aromatic Nitro Precursors into Amines and Synthesis of 3,4-Dihydroquinoxalin-2-Ones

por Iordanidou, Domna, Kallitsakis, Michael G., Tzani, Marina A., Ioannou, Dimitris I., Zarganes-Tzitzikas, Tryfon, Neochoritis, Constantinos G., Dömling, Alexander, Terzidis, Michael A., Lykakis, Ioannis N.
Publicado 2022

Repurposing the HCV NS3–4A protease drug boceprevir as COVID-19 therapeutics

por Oerlemans, Rick, Ruiz-Moreno, Angel Jonathan, Cong, Yingying, Dinesh Kumar, Nilima, Velasco-Velazquez, Marco A., Neochoritis, Constantinos G., Smith, Jolanda, Reggiori, Fulvio, Groves, Matthew R., Dömling, Alexander
Publicado 2020

Optimized Inhibitors of MDM2 via an Attempted Protein‐Templated Reductive Amination

por van der Vlag, Ramon, Yagiz Unver, M., Felicetti, Tommaso, Twarda‐Clapa, Aleksandra, Kassim, Fatima, Ermis, Cagdas, Neochoritis, Constantinos G., Musielak, Bogdan, Labuzek, Beata, Dömling, Alexander, Holak, Tad A., Hirsch, Anna K. H.
Publicado 2019

Rapid approach to complex boronic acids

por Neochoritis, Constantinos G., Shaabani, Shabnam, Ahmadianmoghaddam, Maryam, Zarganes-Tzitzikas, Tryfon, Gao, Li, Novotná, Michaela, Mitríková, Tatiana, Romero, Atilio Reyes, Irianti, Marina Ika, Xu, Ruixue, Olechno, Joe, Ellson, Richard, Helan, Victoria, Kossenjans, Michael, Groves, Matthew R., Dömling, Alexander
Publicado 2019

Design, Synthesis, and Biological Evaluation of 2-Hydroxy-4-phenylthiophene-3-carbonitrile as PD-L1 Antagonist and Its Comparison to Available Small Molecular PD-L1 Inhibitors

por Ważyńska, Marta A., Butera, Roberto, Requesens, Marta, Plat, Annechien, Zarganes-Tzitzikas, Tryfon, Neochoritis, Constantinos G., Plewka, Jacek, Skalniak, Lukasz, Kocik-Krol, Justyna, Musielak, Bogdan, Magiera-Mularz, Katarzyna, Rodriguez, Ismael, Blok, Simon N., de Bruyn, Marco, Nijman, Hans W., Elsinga, Philip H., Holak, Tad A., Dömling, Alexander
Publicado 2023

TEAD–YAP Interaction Inhibitors and MDM2 Binders from DNA‐Encoded Indole‐Focused Ugi Peptidomimetics

por Kunig, Verena B. K., Potowski, Marco, Akbarzadeh, Mohammad, Klika Škopić, Mateja, dos Santos Smith, Denise, Arendt, Lukas, Dormuth, Ina, Adihou, Hélène, Andlovic, Blaž, Karatas, Hacer, Shaabani, Shabnam, Zarganes‐Tzitzikas, Tryfon, Neochoritis, Constantinos G., Zhang, Ran, Groves, Matthew, Guéret, Stéphanie M., Ottmann, Christian, Rahnenführer, Jörg, Fried, Roland, Dömling, Alexander, Brunschweiger, Andreas
Publicado 2020