Design, synthesis, in vitro inhibition and toxicological evaluation of human carbonic anhydrases I, II and IX inhibitors in 5-nitroimidazole series

por Aspatwar, Ashok, Parvathaneni, Nanda Kumar, Barker, Harlan, Anduran, Emilie, Supuran, Claudiu T., Dubois, Ludwig, Lambin, Philippe, Parkkila, Seppo, Winum, Jean-Yves
Publicado 2019

Hypoxia-Activated Prodrug Derivatives of Carbonic Anhydrase Inhibitors in Benzenesulfonamide Series: Synthesis and Biological Evaluation

por Anduran, Emilie, Aspatwar, Ashok, Parvathaneni, Nanda-Kumar, Suylen, Dennis, Bua, Silvia, Nocentini, Alessio, Parkkila, Seppo, Supuran, Claudiu T., Dubois, Ludwig, Lambin, Philippe, Winum, Jean-Yves
Publicado 2020

Nitroimidazole-based inhibitors DTP338 and DTP348 are safe for zebrafish embryos and efficiently inhibit the activity of human CA IX in Xenopus oocytes

por Aspatwar, Ashok, Becker, Holger M., Parvathaneni, Nanda Kumar, Hammaren, Milka, Svorjova, Aleksandra, Barker, Harlan, Supuran, Claudiu T., Dubois, Ludwig, Lambin, Philippe, Parikka, Mataleena, Parkkila, Seppo, Winum, Jean-Yves
Publicado 2018