Covalent Allosteric Inhibitors of Akt Generated Using a Click Fragment Approach

por van der Westhuizen, Leandi, Weisner, Jörn, Taher, Abu, Landel, Ina, Quambusch, Lena, Lindemann, Marius, Uhlenbrock, Niklas, Müller, Matthias P., Green, Ivan R., Pelly, Stephen C., Rauh, Daniel, van Otterlo, Willem A. L.
Publicado 2022

Design and Optimization of Novel Competitive, Non-peptidic, SARS-CoV-2 M(pro) Inhibitors

por Jacobs, Leon, van der Westhuyzen, Aletta, Pribut, Nicole, Dentmon, Zackery W., Cui, Dan, D’Erasmo, Michael P., Bartsch, Perry W., Liu, Ken, Cox, Robert M., Greenlund, Sujay F., Plemper, Richard K., Mitchell, Deborah, Marlow, Joshua, Andrews, Meghan K., Krueger, Rebecca E., Sticher, Zachary M., Kolykhalov, Alexander A., Natchus, Michael G., Zhou, Bin, Pelly, Stephen C., Liotta, Dennis C.
Publicado 2023