2-acetylphenol analogs as potent reversible monoamine oxidase inhibitors

por Legoabe, Lesetja J, Petzer, Anél, Petzer, Jacobus P
Publicado 2015

The Design and Evaluation of an l-Dopa–Lazabemide Prodrug for the Treatment of Parkinson’s Disease

por Hoon, Monique, Petzer, Jacobus P., Viljoen, Francois, Petzer, Anél
Publicado 2017

3-Coumaranone derivatives as inhibitors of monoamine oxidase

por Van Dyk, Adriaan S, Petzer, Jacobus P, Petzer, Anél, Legoabe, Lesetja J
Publicado 2015

Design, synthesis and evaluation of 3-hydroxypyridin-4-ones as inhibitors of catechol-O-methyltransferase

por de Beer, Johannie, Petzer, Jacobus P., Lourens, Anna C. U., Petzer, Anél
Publicado 2020

The evaluation of 1-tetralone and 4-chromanone derivatives as inhibitors of monoamine oxidase

por Cloete, Stephanus J., N’Da, Clarina I., Legoabe, Lesetja J., Petzer, Anél, Petzer, Jacobus P.
Publicado 2020

Coumarin-Based Dual Inhibitors of Human Carbonic Anhydrases and Monoamine Oxidases Featuring Amino Acyl and (Pseudo)-Dipeptidyl Appendages: In Vitro and Computational Studies

por Agamennone, Mariangela, Fantacuzzi, Marialuigia, Carradori, Simone, Petzer, Anél, Petzer, Jacobus P., Angeli, Andrea, Supuran, Claudiu T., Luisi, Grazia
Publicado 2022

Design, Synthesis, Docking Studies and Monoamine Oxidase Inhibition of a Small Library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazoles

por Guglielmi, Paolo, Carradori, Simone, Poli, Giulio, Secci, Daniela, Cirilli, Roberto, Rotondi, Giulia, Chimenti, Paola, Petzer, Anél, Petzer, Jacobus P.
Publicado 2019

SAR and molecular mechanism studies of monoamine oxidase inhibition by selected chalcone analogs

por Shalaby, Raed, Petzer, Jacobus P., Petzer, Anél, Ashraf, Usman M., Atari, Ealla, Alasmari, Fawaz, Kumarasamy, Sivarajan, Sari, Youssef, Khalil, Ashraf
Publicado 2019

4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis

por Secci, Daniela, Carradori, Simone, Petzer, Anél, Guglielmi, Paolo, D’Ascenzio, Melissa, Chimenti, Paola, Bagetta, Donatella, Alcaro, Stefano, Zengin, Gokhan, Petzer, Jacobus P., Ortuso, Francesco
Publicado 2019

Resveratrol Analogues as Dual Inhibitors of Monoamine Oxidase B and Carbonic Anhydrase VII: A New Multi-Target Combination for Neurodegenerative Diseases?

por Carradori, Simone, Fantacuzzi, Marialuigia, Ammazzalorso, Alessandra, Angeli, Andrea, De Filippis, Barbara, Galati, Salvatore, Petzer, Anél, Petzer, Jacobus P., Poli, Giulio, Tuccinardi, Tiziano, Agamennone, Mariangela, Supuran, Claudiu T.
Publicado 2022

Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity

por Guglielmi, Paolo, Secci, Daniela, Petzer, Anél, Bagetta, Donatella, Chimenti, Paola, Rotondi, Giulia, Ferrante, Claudio, Recinella, Lucia, Leone, Sheila, Alcaro, Stefano, Zengin, Gokhan, Petzer, Jacobus P., Ortuso, Francesco, Carradori, Simone
Publicado 2019

Betulin, a Newly Characterized Compound in Acacia auriculiformis Bark, Is a Multi-Target Protein Kinase Inhibitor

por Ahmadu, Augustine A., Delehouzé, Claire, Haruna, Anas, Mustapha, Lukman, Lawal, Bilqis A., Udobre, Aniefiok, Baratte, Blandine, Triscornia, Camilla, Autret, Axelle, Robert, Thomas, Bulinski, Jeannette Chloë, Rousselot, Morgane, Simoes Eugénio, Mélanie, Dimanche-Boitrel, Marie-Thérèse, Petzer, Jacobus P., Legoabe, Lesetja J., Bach, Stéphane
Publicado 2021