A combined fragment-based virtual screening and STD-NMR approach for the identification of E-cadherin ligands

por Vasile, Francesca, Lavore, Francesca, Gazzola, Silvia, Vettraino, Chiara, Parisini, Emilio, Piarulli, Umberto, Belvisi, Laura, Civera, Monica
Publicado 2022

Investigating the Interaction of Cyclic RGD Peptidomimetics with α(V)β(6) Integrin by Biochemical and Molecular Docking Studies

por Civera, Monica, Arosio, Daniela, Bonato, Francesca, Manzoni, Leonardo, Pignataro, Luca, Zanella, Simone, Gennari, Cesare, Piarulli, Umberto, Belvisi, Laura
Publicado 2017

Effects of a novel cyclic RGD peptidomimetic on cell proliferation, migration and angiogenic activity in human endothelial cells

por Fanelli, Roberto, Schembri, Laura, Piarulli, Umberto, Pinoli, Monica, Rasini, Emanuela, Paolillo, Mayra, Galiazzo, Marisa Carlotta, Cosentino, Marco, Marino, Franca
Publicado 2014

Insights into the Binding of Cyclic RGD Peptidomimetics to α(5)β(1) Integrin by using Live‐Cell NMR And Computational Studies

por Guzzetti, Ileana, Civera, Monica, Vasile, Francesca, Arosio, Daniela, Tringali, Cristina, Piarulli, Umberto, Gennari, Cesare, Pignataro, Luca, Belvisi, Laura, Potenza, Donatella
Publicado 2016

Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting

por Bodero, Lizeth, López Rivas, Paula, Korsak, Barbara, Hechler, Torsten, Pahl, Andreas, Müller, Christoph, Arosio, Daniela, Pignataro, Luca, Gennari, Cesare, Piarulli, Umberto
Publicado 2018

Cyclic RGD and isoDGR Integrin Ligands Containing cis-2-amino-1-cyclopentanecarboxylic (cis-β-ACPC) Scaffolds

por Panzeri, Silvia, Arosio, Daniela, Gazzola, Silvia, Belvisi, Laura, Civera, Monica, Potenza, Donatella, Vasile, Francesca, Kemker, Isabell, Ertl, Thomas, Sewald, Norbert, Reiser, Oliver, Piarulli, Umberto
Publicado 2020

Synthesis and Biological Evaluation of RGD and isoDGR–Monomethyl Auristatin Conjugates Targeting Integrin α(V)β(3)

por Raposo Moreira Dias, André, Bodero, Lizeth, Martins, Ana, Arosio, Daniela, Gazzola, Silvia, Belvisi, Laura, Pignataro, Luca, Steinkühler, Christian, Dal Corso, Alberto, Gennari, Cesare, Piarulli, Umberto
Publicado 2019

Conformational switch and multiple supramolecular structures of a newly identified self-assembling protein-mimetic peptide from Pseudomonas aeruginosa YeaZ protein

por Fasola, Elettra, Alboreggia, Giulia, Pieraccini, Stefano, Oliva, Francesco, Agharbaoui, Fatima Ezzahra, Bollati, Michela, Bertoni, Giovanni, Recchia, Sandro, Marelli, Marcello, Piarulli, Umberto, Pellegrino, Sara, Gazzola, Silvia
Publicado 2022

Optimizing the enzymatic release of MMAE from isoDGR-based small molecule drug conjugate by incorporation of a GPLG-PABC enzymatically cleavable linker

por Zambra, Marco, Ranđelović, Ivan, Talarico, Francesco, Borbély, Adina, Svajda, Laura, Tóvári, József, Mező, Gábor, Bodero, Lizeth, Colombo, Sveva, Arrigoni, Federico, Fasola, Elettra, Gazzola, Silvia, Piarulli, Umberto
Publicado 2023

Synthesis, Characterization, and Biological Evaluation of a Dual-Action Ligand Targeting α(v)β(3) Integrin and VEGF Receptors**

por Zanella, Simone, Mingozzi, Michele, Dal Corso, Alberto, Fanelli, Roberto, Arosio, Daniela, Cosentino, Marco, Schembri, Laura, Marino, Franca, De Zotti, Marta, Formaggio, Fernando, Pignataro, Luca, Belvisi, Laura, Piarulli, Umberto, Gennari, Cesare
Publicado 2015

Rational Design of Antiangiogenic Helical Oligopeptides Targeting the Vascular Endothelial Growth Factor Receptors

por Zanella, Simone, Bocchinfuso, Gianfranco, De Zotti, Marta, Arosio, Daniela, Marino, Franca, Raniolo, Stefano, Pignataro, Luca, Sacco, Giovanni, Palleschi, Antonio, Siano, Alvaro S., Piarulli, Umberto, Belvisi, Laura, Formaggio, Fernando, Gennari, Cesare, Stella, Lorenzo
Publicado 2019

Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery

por Borbély, Adina, Figueras, Eduard, Martins, Ana, Bodero, Lizeth, Raposo Moreira Dias, André, López Rivas, Paula, Pina, Arianna, Arosio, Daniela, Gallinari, Paola, Frese, Marcel, Steinkühler, Christian, Gennari, Cesare, Piarulli, Umberto, Sewald, Norbert
Publicado 2019

Tumor Targeting with an isoDGR–Drug Conjugate

por Zanella, Simone, Angerani, Simona, Pina, Arianna, López Rivas, Paula, Giannini, Clelia, Panzeri, Silvia, Arosio, Daniela, Caruso, Michele, Gasparri, Fabio, Fraietta, Ivan, Albanese, Clara, Marsiglio, Aurelio, Pignataro, Luca, Belvisi, Laura, Piarulli, Umberto, Gennari, Cesare
Publicado 2017