Evaluation of Ruthenium(II) N-Heterocyclic Carbene Complexes as Antibacterial Agents and Inhibitors of Bacterial Thioredoxin Reductase

por Burmeister, Hilke, Dietze, Pascal, Preu, Lutz, Bandow, Julia E., Ott, Ingo
Publicado 2021

Novel 2-Phenoxyanilide Congeners Derived from a Hit Structure of the TCAMS: Synthesis and Evaluation of Their in Vitro Activity against Plasmodium falciparum

por Weidner, Thomas, Nasereddin, Abed, Preu, Lutz, Grünefeld, Johann, Dzikowski, Ron, Kunick, Conrad
Publicado 2016

Indole-3-Carbonitriles as DYRK1A Inhibitors by Fragment-Based Drug Design

por Meine, Rosanna, Becker, Walter, Falke, Hannes, Preu, Lutz, Loaëc, Nadège, Meijer, Laurent, Kunick, Conrad
Publicado 2018

Antiplasmodial dihetarylthioethers target the coenzyme A synthesis pathway in Plasmodium falciparum erythrocytic stages

por Weidner, Thomas, Lucantoni, Leonardo, Nasereddin, Abed, Preu, Lutz, Jones, Peter G., Dzikowski, Ron, Avery, Vicky M., Kunick, Conrad
Publicado 2017

Molecular structures of cdc2-like kinases in complex with a new inhibitor chemotype

por Walter, Anne, Chaikuad, Apirat, Helmer, Renate, Loaëc, Nadège, Preu, Lutz, Ott, Ingo, Knapp, Stefan, Meijer, Laurent, Kunick, Conrad
Publicado 2018

[b]-Annulated Halogen-Substituted Indoles as Potential DYRK1A Inhibitors

por Lechner, Christian, Flaßhoff, Maren, Falke, Hannes, Preu, Lutz, Loaëc, Nadége, Meijer, Laurent, Knapp, Stefan, Chaikuad, Apirat, Kunick, Conrad
Publicado 2019

Structure–activity relationships in a series of antiplasmodial thieno[2,3-b]pyridines

por Masch, Andreas, Nasereddin, Abed, Alder, Arne, Bird, Megan J., Schweda, Sandra I., Preu, Lutz, Doerig, Christian, Dzikowski, Ron, Gilberger, Tim W., Kunick, Conrad
Publicado 2019

10-Iodo-11H-indolo[3,2-c]quinoline-6-carboxylic Acids Are Selective Inhibitors of DYRK1A

por Falke, Hannes, Chaikuad, Apirat, Becker, Anja, Loaëc, Nadège, Lozach, Olivier, Abu Jhaisha, Samira, Becker, Walter, Jones, Peter G., Preu, Lutz, Baumann, Knut, Knapp, Stefan, Meijer, Laurent, Kunick, Conrad
Publicado 2015