One-pot multicomponent green Hantzsch synthesis of 1,2-dihydropyridine derivatives with antiproliferative activity

por Bosica, Giovanna, Demanuele, Kaylie, Padrón, José M, Puerta, Adrián
Publicado 2020

Correction: One-pot multicomponent green Hantzsch synthesis of 1,2-dihydropyridine derivatives with antiproliferative activity

por Bosica, Giovanna, Demanuele, Kaylie, Padrón, José Manuel, Puerta, Adrián
Publicado 2021

Early Pharmacological Profiling of Antiproliferative Compounds by Live Cell Imaging

por Puerta, Adrián, González-Bakker, Aday, Santos, Guido, Padrón, José M.
Publicado 2022

Alkaloid Profiling, Anti-Enzymatic and Antiproliferative Activity of the Endemic Chilean Amaryllidaceae Phycella cyrtanthoides

por Fernández-Galleguillos, Carlos, Romero-Parra, Javier, Puerta, Adrián, Padrón, José M., Simirgiotis, Mario J.
Publicado 2022

UHPLC-MS Chemical Fingerprinting and Antioxidant, Antiproliferative, and Enzyme Inhibition Potential of Gaultheria pumila Berries

por Fernández-Galleguillos, Carlos, Quesada-Romero, Luisa, Puerta, Adrián, Padrón, José M., Souza, Ernane, Romero-Parra, Javier, Simirgiotis, Mario J.
Publicado 2021

A New Oxadiazole-Based Topsentin Derivative Modulates Cyclin-Dependent Kinase 1 Expression and Exerts Cytotoxic Effects on Pancreatic Cancer Cells

por Pecoraro, Camilla, Parrino, Barbara, Cascioferro, Stella, Puerta, Adrian, Avan, Amir, Peters, Godefridus J., Diana, Patrizia, Giovannetti, Elisa, Carbone, Daniela
Publicado 2021

New Pharmacological Strategies against Pancreatic Adenocarcinoma: The Multifunctional Thiosemicarbazone FA4

por Anobile, Dario P., Niso, Mauro, Puerta, Adrian, Fraga Rodrigues, Stephanie M., Abatematteo, Francesca S., Avan, Amir, Abate, Carmen, Riganti, Chiara, Giovannetti, Elisa
Publicado 2022

Investigation of the enantioselectivity of acetylcholinesterase and butyrylcholinesterase upon inhibition by tacrine-iminosugar heterodimers

por Vaaland, I. Caroline, López, Óscar, Puerta, Adrián, Fernandes, Miguel X., Padrón, José M., Fernández-Bolaños, José G., Sydnes, Magne O., Lindbäck, Emil
Publicado 2022

Synthesis and Evaluation of Pyrimidine Steroids as Antiproliferative Agents

por Cortés-Percino, Alejandra, Vega-Báez, José Luis, Romero-López, Anabel, Puerta, Adrián, Merino-Montiel, Penélope, Meza-Reyes, Socorro, Padrón, José M., Montiel-Smith, Sara
Publicado 2019

Masked Phenolic-Selenium Conjugates: Potent and Selective Antiproliferative Agents Overcoming P-gp Resistance

por Begines, Paloma, Sevilla-Horrillo, Lucía, Puerta, Adrián, Puckett, Rebecca, Bayort, Samuel, Lagunes, Irene, Maya, Inés, Padrón, José M., López, Óscar, Fernández-Bolaños, José G.
Publicado 2020

Phenolic Fingerprinting and Bioactivity Profiling of Extracts and Isolated Compounds from Gypothamnium pinifolium Phil.

por Barrientos, Ruth E., Ibáñez, Elena, Puerta, Adrián, Padrón, José M., Paredes, Adrián, Cifuentes, Fredi, Romero-Parra, Javier, Palacios, Javier, Bórquez, Jorge, Simirgiotis, Mario J.
Publicado 2022

Squaramide-Tethered Sulfonamides and Coumarins: Synthesis, Inhibition of Tumor-Associated CAs IX and XII and Docking Simulations

por Arrighi, Giulia, Puerta, Adrián, Petrini, Andrea, Hicke, Francisco J., Nocentini, Alessio, Fernandes, Miguel X., Padrón, José M., Supuran, Claudiu T., Fernández-Bolaños, José G., López, Óscar
Publicado 2022

Bioactive Potential: A Pharmacognostic Definition through the Screening of Four Hypericum Species from the Canary Islands

por Lacret, Rodney, Puerta, Adrián, Granica, Sebastian, González-Bakker, Aday, Hevia, Danela, Teng, Yiling, Sánchez-Mateo, Candelaria C., Pérez de Paz, Pedro Luis, Padrón, José M.
Publicado 2022

Microwave-assisted multicomponent synthesis of antiproliferative 2,4-dimethoxy-tetrahydropyrimido[4,5-b]quinolin-6(7H)-ones

por Patel, Subham G., González-Bakker, Aday, Vala, Ruturajsinh M., Patel, Paras J., Puerta, Adrián, Malik, Apoorva, Sharma, Rakesh K., Padrón, José M., Patel, Hitendra M.
Publicado 2022

A hybrid of 1-deoxynojirimycin and benzotriazole induces preferential inhibition of butyrylcholinesterase (BuChE) over acetylcholinesterase (AChE)

por Evangelista, Tereza Cristina Santos, López, Óscar, Puerta, Adrián, Fernandes, Miguel X., Ferreira, Sabrina Baptista, Padrón, José M., Fernández-Bolaños, José G., Sydnes, Magne O., Lindbäck, Emil
Publicado 2022

Oxonitrogenated Derivatives of Eremophilans and Eudesmans: Antiproliferative and Anti-Trypanosoma cruzi Activity

por Beer, María F., Reta, Guillermo F., Puerta, Adrián, Bivona, Augusto E., Alberti, Andrés Sánchez, Cerny, Natacha, Malchiodi, Emilio L., Tonn, Carlos E., Padrón, José M., Sülsen, Valeria P., Donadel, Osvaldo J.
Publicado 2022

2-Aminobenzoxazole-appended coumarins as potent and selective inhibitors of tumour-associated carbonic anhydrases

por Fuentes-Aguilar, Alma, Merino-Montiel, Penélope, Montiel-Smith, Sara, Meza-Reyes, Socorro, Vega-Báez, José Luis, Puerta, Adrián, Fernandes, Miguel X., Padrón, José M., Petreni, Andrea, Nocentini, Alessio, Supuran, Claudiu T., López, Óscar, Fernández-Bolaños, José G.
Publicado 2021

Conformationally Restricted Glycoconjugates Derived from Arylsulfonamides and Coumarins: New Families of Tumour-Associated Carbonic Anhydrase Inhibitors

por Martínez-Montiel, Mónica, Romero-Hernández, Laura L., Giovannuzzi, Simone, Begines, Paloma, Puerta, Adrián, Ahuja-Casarín, Ana I., Fernandes, Miguel X., Merino-Montiel, Penélope, Montiel-Smith, Sara, Nocentini, Alessio, Padrón, José M., Supuran, Claudiu T., Fernández-Bolaños, José G., López, Óscar
Publicado 2023

A Comprehensive Evaluation of Sdox, a Promising H(2)S-Releasing Doxorubicin for the Treatment of Chemoresistant Tumors

por Alov, Petko, Al Sharif, Merilin, Aluani, Denitsa, Chegaev, Konstantin, Dinic, Jelena, Divac Rankov, Aleksandra, Fernandes, Miguel X., Fusi, Fabio, García-Sosa, Alfonso T., Juvonen, Risto, Kondeva-Burdina, Magdalena, Padrón, José M., Pajeva, Ilza, Pencheva, Tania, Puerta, Adrián, Raunio, Hannu, Riganti, Chiara, Tsakovska, Ivanka, Tzankova, Virginia, Yordanov, Yordan, Saponara, Simona
Publicado 2022