Structure–Activity Relationships (SARs) of α-Ketothioamides as Inhibitors of Phosphoglycerate Dehydrogenase (PHGDH)

por Spillier, Quentin, Ravez, Séverine, Unterlass, Judith, Corbet, Cyril, Degavre, Charline, Feron, Olivier, Frédérick, Raphaël
Publicado 2020

Unravelling the Allosteric Targeting of PHGDH at the ACT-Binding Domain with a Photoactivatable Diazirine Probe and Mass Spectrometry Experiments †

por Spillier, Quentin, Ravez, Séverine, Dochain, Simon, Vertommen, Didier, Thabault, Léopold, Feron, Olivier, Frédérick, Raphaël
Publicado 2021

Anti-alcohol abuse drug disulfiram inhibits human PHGDH via disruption of its active tetrameric form through a specific cysteine oxidation

por Spillier, Quentin, Vertommen, Didier, Ravez, Séverine, Marteau, Romain, Thémans, Quentin, Corbet, Cyril, Feron, Olivier, Wouters, Johan, Frédérick, Raphaël
Publicado 2019

MUC4-ErbB2 Oncogenic Complex: Binding studies using Microscale Thermophoresis

por Liberelle, Maxime, Magnez, Romain, Thuru, Xavier, Bencheikh, Yamina, Ravez, Severine, Quenon, Camille, Drucbert, Anne-Sophie, Foulon, Catherine, Melnyk, Patricia, Seuningen, Isabelle Van, Lebègue, Nicolas
Publicado 2019

Publisher Correction: MUC4-ErbB2 Oncogenic Complex: Binding studies using Microscale Thermophoresis

por Liberelle, Maxime, Magnez, Romain, Thuru, Xavier, Bencheikh, Yamina, Ravez, Severine, Quenon, Camille, Drucbert, Anne-Sophie, Foulon, Catherine, Melnyk, Patricia, Van Seuningen, Isabelle, Lebègue, Nicolas
Publicado 2020

Safe and Efficient Sigma1 Ligand: A Potential Drug Candidate for Multiple Sclerosis

por Oxombre, Bénédicte, Madouri, Fahima, Journé, Anne-Sophie, Ravez, Séverine, Woitrain, Eloise, Odou, Pascal, Duhal, Nathalie, Ninni, Sandro, Montaigne, David, Delhem, Nadira, Vermersch, Patrick, Melnyk, Patricia
Publicado 2022