Design, Synthesis and Characterization of a New Series of Fluorescent Metabotropic Glutamate Receptor Type 5 Negative Allosteric Modulators

por Fernández-Dueñas, Víctor, Qian, Mingcheng, Argerich, Josep, Amaral, Carolina, Risseeuw, Martijn D.P., Van Calenbergh, Serge, Ciruela, Francisco
Publicado 2020

Synthesis of Extended Uridine Phosphonates Derived from an Allosteric P2Y(2) Receptor Ligand

por Song, Lijun, Risseeuw, Martijn D. P., Karalic, Izet, Barrett, Matthew O., Brown, Kyle A., Harden, T. Kendall, Van Calenbergh, Serge
Publicado 2014

Synthetic Fosmidomycin Analogues with Altered Chelating Moieties Do Not Inhibit 1-Deoxy-d-xylulose 5-phosphate Reductoisomerase or Plasmodium falciparum Growth In Vitro

por Chofor, René, Risseeuw, Martijn D.P., Pouyez, Jenny, Johny, Chinchu, Wouters, Johan, Dowd, Cynthia S., Couch, Robin D., Van Calenbergh, Serge
Publicado 2014

1-(Piperidin-3-yl)thymine amides as inhibitors of M. tuberculosis thymidylate kinase

por Jian, Yanlin, Risseeuw, Martijn D. P., Froeyen, Mathy, Song, Lijun, Cappoen, Davie, Cos, Paul, Munier-Lehmann, Hélène, van Calenbergh, Serge
Publicado 2019

Mucosal and blood-brain barrier transport kinetics of the plant N-alkylamide spilanthol using in vitro and in vivo models

por Veryser, Lieselotte, Taevernier, Lien, Joshi, Tanmayee, Tatke, Pratima, Wynendaele, Evelien, Bracke, Nathalie, Stalmans, Sofie, Peremans, Kathelijne, Burvenich, Christian, Risseeuw, Martijn, De Spiegeleer, Bart
Publicado 2016

1-(1-Arylethylpiperidin-4-yl)thymine Analogs as Antimycobacterial TMPK Inhibitors

por Jian, Yanlin, Hulpia, Fabian, D. P. Risseeuw, Martijn, Forbes, He Eun, Caljon, Guy, Munier-Lehmann, Hélène, I. M. Boshoff, Helena, Van Calenbergh, Serge
Publicado 2020

Host metabolites stimulate the bacterial proton motive force to enhance the activity of aminoglycoside antibiotics

por Crabbé, Aurélie, Ostyn, Lisa, Staelens, Sorien, Rigauts, Charlotte, Risseeuw, Martijn, Dhaenens, Maarten, Daled, Simon, Van Acker, Heleen, Deforce, Dieter, Van Calenbergh, Serge, Coenye, Tom
Publicado 2019

Galactosylsphingamides: new α-GalCer analogues to probe the F’-pocket of CD1d

por Guillaume, Joren, Wang, Jing, Janssens, Jonas, Remesh, Soumya G., Risseeuw, Martijn D. P., Decruy, Tine, Froeyen, Mathy, Elewaut, Dirk, Zajonc, Dirk M., Calenbergh, Serge Van
Publicado 2017

A “Clickable” MTX Reagent as a Practical Tool for Profiling Small-Molecule–Intracellular Target Interactions via MASPIT

por Risseeuw, Martijn D P, De Clercq, Dries J H, Lievens, Sam, Hillaert, Ulrik, Sinnaeve, Davy, Van den Broeck, Freya, Martins, José C, Tavernier, Jan, Van Calenbergh, Serge
Publicado 2013