Amino Acids as Building Blocks for Carbonic Anhydrase Inhibitors

por Chiaramonte, Niccolò, Romanelli, Maria Novella, Teodori, Elisabetta, Supuran, Claudiu T.
Publicado 2018

Recent advances in the search of BCRP- and dual P-gp/BCRP-based multidrug resistance modulators

por Dei, Silvia, Braconi, Laura, Romanelli, Maria Novella, Teodori, Elisabetta
Publicado 2019

Effectiveness of the Histone Deacetylase Inhibitor (S)-2 against LNCaP and PC3 Human Prostate Cancer Cells

por Laurenzana, Anna, Balliu, Manjola, Cellai, Cristina, Romanelli, Maria Novella, Paoletti, Francesco
Publicado 2013

Investigation of piperazines as human carbonic anhydrase I, II, IV and VII activators

por Angeli, Andrea, Chiaramonte, Niccolò, Manetti, Dina, Romanelli, Maria Novella, Supuran, Claudiu T.
Publicado 2017

Dual HDAC/BRD4 Inhibitors Relieves Neuropathic Pain by Attenuating Inflammatory Response in Microglia After Spared Nerve Injury

por Borgonetti, Vittoria, Meacci, Elisabetta, Pierucci, Federica, Romanelli, Maria Novella, Galeotti, Nicoletta
Publicado 2022

HDAC-inhibitor (S)-8 disrupts HDAC6-PP1 complex prompting A375 melanoma cell growth arrest and apoptosis

por Balliu, Manjola, Guandalini, Luca, Romanelli, Maria Novella, D'Amico, Massimo, Paoletti, Francesco
Publicado 2015

HCN Channels Modulators: The Need for Selectivity

por Romanelli, Maria Novella, Sartiani, Laura, Masi, Alessio, Mannaioni, Guido, Manetti, Dina, Mugelli, Alessandro, Cerbai, Elisabetta
Publicado 2016

Recent Advances in the Discovery of Nicotinic Acetylcholine Receptor Allosteric Modulators

por Manetti, Dina, Dei, Silvia, Arias, Hugo R., Braconi, Laura, Gabellini, Alessio, Teodori, Elisabetta, Romanelli, Maria Novella
Publicado 2023

New Histamine-Related Five-Membered N-Heterocycle Derivatives as Carbonic Anhydrase I Activators

por Chiaramonte, Niccolò, Gabellini, Alessio, Angeli, Andrea, Bartolucci, Gianluca, Braconi, Laura, Dei, Silvia, Teodori, Elisabetta, Supuran, Claudiu T., Romanelli, Maria Novella
Publicado 2022

Two types of interneurons in the mouse lateral geniculate nucleus are characterized by different h-current density

por Leist, Michael, Datunashvilli, Maia, Kanyshkova, Tatyana, Zobeiri, Mehrnoush, Aissaoui, Ania, Cerina, Manuela, Romanelli, Maria Novella, Pape, Hans-Christian, Budde, Thomas
Publicado 2016

A potentiated cooperation of carbonic anhydrase IX and histone deacetylase inhibitors against cancer

por Ruzzolini, Jessica, Laurenzana, Anna, Andreucci, Elena, Peppicelli, Silvia, Bianchini, Francesca, Carta, Fabrizio, Supuran, Claudiu T., Romanelli, Maria Novella, Nediani, Chiara, Calorini, Lido
Publicado 2019

Dual P-Glycoprotein and CA XII Inhibitors: A New Strategy to Reverse the P-gp Mediated Multidrug Resistance (MDR) in Cancer Cells †

por Teodori, Elisabetta, Braconi, Laura, Bua, Silvia, Lapucci, Andrea, Bartolucci, Gianluca, Manetti, Dina, Romanelli, Maria Novella, Dei, Silvia, Supuran, Claudiu T., Coronnello, Marcella
Publicado 2020

Synthesis and carbonic anhydrase activating properties of a series of 2-amino-imidazolines structurally related to clonidine(1)

por Chiaramonte, Niccolò, Maach, Soumia, Biliotti, Caterina, Angeli, Andrea, Bartolucci, Gianluca, Braconi, Laura, Dei, Silvia, Teodori, Elisabetta, Supuran, Claudiu T., Romanelli, Maria Novella
Publicado 2020

Evaluating the efficiency of enzyme accelerated CO(2) capture: chemical kinetics modelling for interpreting measurement results

por Parri, Lorenzo, Fort, Ada, Lo Grasso, Anna, Mugnaini, Marco, Vignoli, Valerio, Capasso, Clemente, Del Prete, Sonia, Romanelli, Maria Novella, Supuran, Claudiu T.
Publicado 2021

The Antinociceptive Activity of (E)-3-(thiophen-2-yl)-N-(p-tolyl)acrylamide in Mice Is Reduced by (E)-3-(furan-2-yl)-N-methyl-N-(p-tolyl)acrylamide Through Opposing Modulatory Mech...

por Arias, Hugo R., Tae, Han-Shen, Micheli, Laura, Yousuf, Arsalan, Manetti, Dina, Romanelli, Maria Novella, Ghelardini, Carla, Adams, David J., Di Cesare Mannelli, Lorenzo
Publicado 2023

Overcoming Multidrug Resistance (MDR): Design, Biological Evaluation and Molecular Modelling Studies of 2,4‐Substituted Quinazoline Derivatives

por Braconi, Laura, Teodori, Elisabetta, Contino, Marialessandra, Riganti, Chiara, Bartolucci, Gianluca, Manetti, Dina, Romanelli, Maria Novella, Perrone, Maria Grazia, Colabufo, Nicola Antonio, Guglielmo, Stefano, Dei, Silvia
Publicado 2022

New Dual P-Glycoprotein (P-gp) and Human Carbonic Anhydrase XII (hCA XII) Inhibitors as Multidrug Resistance (MDR) Reversers in Cancer Cells

por Braconi, Laura, Teodori, Elisabetta, Riganti, Chiara, Coronnello, Marcella, Nocentini, Alessio, Bartolucci, Gianluca, Pallecchi, Marco, Contino, Marialessandra, Manetti, Dina, Romanelli, Maria Novella, Supuran, Claudiu T., Dei, Silvia
Publicado 2022

6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers

por Braconi, Laura, Bartolucci, Gianluca, Contino, Marialessandra, Chiaramonte, Niccolò, Giampietro, Roberta, Manetti, Dina, Perrone, Maria Grazia, Romanelli, Maria Novella, Colabufo, Nicola Antonio, Riganti, Chiara, Dei, Silvia, Teodori, Elisabetta
Publicado 2020

Selective Blockade of HCN1/HCN2 Channels as a Potential Pharmacological Strategy Against Pain

por Dini, Leonardo, Del Lungo, Martina, Resta, Francesco, Melchiorre, Michele, Spinelli, Valentina, Di Cesare Mannelli, Lorenzo, Ghelardini, Carla, Laurino, Annunziatina, Sartiani, Laura, Coppini, Raffaele, Mannaioni, Guido, Cerbai, Elisabetta, Romanelli, Maria Novella
Publicado 2018

Carbonic Anhydrase IV Selective Inhibitors Counteract the Development of Colitis-Associated Visceral Pain in Rats

por Lucarini, Elena, Nocentini, Alessio, Bonardi, Alessandro, Chiaramonte, Niccolò, Parisio, Carmen, Micheli, Laura, Toti, Alessandra, Ferrara, Valentina, Carrino, Donatello, Pacini, Alessandra, Romanelli, Maria Novella, Supuran, Claudiu T., Ghelardini, Carla, Di Cesare Mannelli, Lorenzo
Publicado 2021