Design, Synthesis, Docking Studies and Monoamine Oxidase Inhibition of a Small Library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazoles

por Guglielmi, Paolo, Carradori, Simone, Poli, Giulio, Secci, Daniela, Cirilli, Roberto, Rotondi, Giulia, Chimenti, Paola, Petzer, Anél, Petzer, Jacobus P.
Publicado 2019

Discovery, affinity maturation and multimerization of small molecule ligands against human tyrosinase and tyrosinase-related protein 1

por Catalano, Marco, Bassi, Gabriele, Rotondi, Giulia, Khettabi, Lyna, Dichiara, Maria, Murer, Patrizia, Scheuermann, Jörg, Soler-Lopez, Montserrat, Neri, Dario
Publicado 2020

Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation

por Guglielmi, Paolo, Rotondi, Giulia, Secci, Daniela, Angeli, Andrea, Chimenti, Paola, Nocentini, Alessio, Bonardi, Alessandro, Gratteri, Paola, Carradori, Simone, Supuran, Claudiu T.
Publicado 2020

Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold

por Rotondi, Giulia, Guglielmi, Paolo, Carradori, Simone, Secci, Daniela, De Monte, Celeste, De Filippis, Barbara, Maccallini, Cristina, Amoroso, Rosa, Cirilli, Roberto, Akdemir, Atilla, Angeli, Andrea, Supuran, Claudiu T.
Publicado 2019

Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity

por Guglielmi, Paolo, Secci, Daniela, Petzer, Anél, Bagetta, Donatella, Chimenti, Paola, Rotondi, Giulia, Ferrante, Claudio, Recinella, Lucia, Leone, Sheila, Alcaro, Stefano, Zengin, Gokhan, Petzer, Jacobus P., Ortuso, Francesco, Carradori, Simone
Publicado 2019