Pyrimido[1,2-a]benzimidazoles: synthesis and perspective of their pharmacological use

por Fedotov, Victor V., Rusinov, Vladimir L., Ulomsky, Evgeny N., Mukhin, Evgeny M., Gorbunov, Evgeny B., Chupakhin, Oleg N.
Publicado 2021

Oxidative Aromatization of 4,7-Dihydro-6-nitroazolo[1,5-a]pyrimidines: Synthetic Possibilities and Limitations, Mechanism of Destruction, and the Theoretical and Experimental Subst...

por Lyapustin, Daniil N., Ulomsky, Evgeny N., Balyakin, Ilya A., Shchepochkin, Alexander V., Rusinov, Vladimir L., Chupakhin, Oleg N.
Publicado 2021

6-(Tetrazol-5-yl)-7-aminoazolo[1,5-a]pyrimidines as Novel Potent CK2 Inhibitors

por Urakov, Grigoriy V., Savateev, Konstantin V., Kotovskaya, Svetlana K., Rusinov, Vladimir L., Spasov, Alexandr A., Babkov, Denis A., Sokolova, Elena V.
Publicado 2022

Redox Conversions of 5-Methyl-6-nitro-7-oxo-4,7-dihydro-1,2,4triazolo[1,5-a]pyrimidinide L-Arginine Monohydrate as a Promising Antiviral Drug

por Ivoilova, Alexandra, Mikhalchenko, Ludmila V., Tsmokalyuk, Anton, Leonova, Marina, Lalov, Andrey, Mozharovskaia, Polina, Kozitsina, Alisa N., Ivanova, Alla V., Rusinov, Vladimir L.
Publicado 2021

Mechanochemical Approach towards Multi-Functionalized 1,2,3-Triazoles and Anti-Seizure Drug Rufinamide Analogs Using Copper Beads

por Bhattacherjee, Dhananjay, Kovalev, Igor S., Kopchuk, Dmitry S., Rahman, Matiur, Santra, Sougata, Zyryanov, Grigory V., Das, Pralay, Purohit, Rituraj, Rusinov, Vladimir L., Chupakhin, Oleg N.
Publicado 2022

Antiviral drug Triazavirin, selectively labeled with (2)H, (13)C, and (15)N stable isotopes. Synthesis and properties

por Shestakova, Tatyana S., Deev, Sergey L., Khalymbadzha, Igor А., Rusinov, Vladimir L., Paramonov, Alexander S., Arseniev, Alexander S., Shenkarev, Zakhar O., Charushin, Valery N., Chupakhin, Oleg N.
Publicado 2021

Triazavirin—A Novel Effective Antiviral Drug

por Chupakhin, Oleg N., Rusinov, Vladimir L., Varaksin, Mikhail V., Ulomskiy, Evgeny N., Savateev, Konstantin V., Butorin, Ilya I., Du, Weijie, Sun, Zhiyong, Charushin, Valery N.
Publicado 2022

(15)N-Labelling and structure determination of adamantylated azolo-azines in solution

por Deev, Sergey L, Paramonov, Alexander S, Shestakova, Tatyana S, Khalymbadzha, Igor A, Chupakhin, Oleg N, Subbotina, Julia O, Eltsov, Oleg S, Slepukhin, Pavel A, Rusinov, Vladimir L, Arseniev, Alexander S, Shenkarev, Zakhar O
Publicado 2017

Methods of Synthesis and Antiviral Activity of New 4-Alkyl-3-Nitro-1,4-Dihydroazolo[5,1-c][1,2,4]Triazin-4-ols

por Drokin, Roman A., Tiufiakov, Dmitrii V., Voinkov, Egor K., Slepukhin, Pavel A., Ulomsky, Evgeny N., Esaulkova, Yana L., Volobueva, Alexandrina S., Lantseva, Kristina S., Misyurina, Mariya A., Zarubaev, Vladimir V., Rusinov, Vladimir L.
Publicado 2021

Azolo[1,5-a]pyrimidines and Their Condensed Analogs with Anticoagulant Activity

por Savateev, Konstantin V., Fedotov, Victor V., Rusinov, Vladimir L., Kotovskaya, Svetlana K., Spasov, Alexandr A., Kucheryavenko, Aida F., Vasiliev, Pavel M., Kosolapov, Vadim A., Sirotenko, Victor S., Gaidukova, Kseniya A., Uskov, Georgiy M.
Publicado 2022

4-(Aryl)-Benzo[4,5]imidazo[1,2-a]pyrimidine-3-Carbonitrile-Based Fluorophores: Povarov Reaction-Based Synthesis, Photophysical Studies, and DFT Calculations

por Fedotov, Victor V., Valieva, Maria I., Taniya, Olga S., Aminov, Semen V., Kharitonov, Mikhail A., Novikov, Alexander S., Kopchuk, Dmitry S., Slepukhin, Pavel A., Zyryanov, Grigory V., Ulomsky, Evgeny N., Rusinov, Vladimir L., Charushin, Valery N.
Publicado 2022

Aerosol Inhalation Delivery of Triazavirin in Mice: Outlooks for Advanced Therapy Against Novel Viral Infections

por Valiulin, Sergey V., Onischuk, Andrey A., Dubtsov, Sergey N., Baklanov, Anatoly M., An'kov, Sergey V., Plokhotnichenko, Maria E., Tolstikova, Tatyana G., Dultseva, Galina G., Rusinov, Vladimir L., Charushin, Valery N., Fomin, Vasily M.
Publicado 2021

CK2 Inhibition and Antitumor Activity of 4,7-Dihydro-6-nitroazolo[1,5-a]pyrimidines

por Lyapustin, Daniil N., Kotovskaya, Svetlana K., Butorin, Ilya I., Ulomsky, Evgeny N., Rusinov, Vladimir L., Babkov, Denis A., Pokhlebin, Alexander A., Spasov, Alexander A., Melekhin, Vsevolod V., Tokhtueva, Maria D., Shcheglova, Anna V., Makeev, Oleg G.
Publicado 2022