Continuous enzyme activity assay for high-throughput classification of histone deacetylase 8 inhibitors

por Schweipert, Markus, Amurthavasan, Anuja, Meyer-Almes, Franz-Josef
Publicado 2023

Synthesis and HDAC inhibitory activity of pyrimidine-based hydroxamic acids

por Jakubkiene, Virginija, Valiulis, Gabrielius Ernis, Schweipert, Markus, Zubriene, Asta, Matulis, Daumantas, Meyer-Almes, Franz-Josef, Tumkevicius, Sigitas
Publicado 2022

Mechanistic Insights into Binding of Ligands with Thiazolidinedione Warhead to Human Histone Deacetylase 4

por Schweipert, Markus, Jänsch, Niklas, Upadhyay, Neha, Tilekar, Kalpana, Wozny, Ewelina, Basheer, Sidra, Wurster, Eva, Müller, Marlene, C S, Ramaa, Meyer-Almes, Franz-Josef
Publicado 2021

Design, Synthesis, and Biological Evaluation of Novel Quinazolin-4(3H)-One-Based Histone Deacetylase 6 (HDAC6) Inhibitors for Anticancer Activity

por Khetmalis, Yogesh Mahadu, Fathima, Ashna, Schweipert, Markus, Debarnot, Cécile, Bandaru, Naga Venkata Madhusudhan Rao, Murugesan, Sankaranarayanan, Jamma, Trinath, Meyer-Almes, Franz-Josef, Sekhar, Kondapalli Venkata Gowri Chandra
Publicado 2023

3‐Chloro‐5‐Substituted‐1,2,4‐Thiadiazoles (TDZs) as Selective and Efficient Protein Thiol Modifiers

por Jänsch, Niklas, Frühauf, Anton, Schweipert, Markus, Debarnot, Cécile, Erhardt, Miriam, Brenner‐Weiss, Gerald, Kirschhöfer, Frank, Jasionis, Tomas, Čapkauskaitė, Edita, Zubrienė, Asta, Matulis, Daumantas, Meyer‐Almes, Franz‐Josef
Publicado 2022