Structure‐Enabled Discovery of a Stapled Peptide Inhibitor to Target the Oncogenic Transcriptional Repressor TLE1

por McGrath, Sally, Tortorici, Marcello, Drouin, Ludovic, Solanki, Savade, Vidler, Lewis, Westwood, Isaac, Gimeson, Peter, Van Montfort, Rob, Hoelder, Swen
Publicado 2017

Aminopyrazine Inhibitors Binding to an Unusual Inactive Conformation of the Mitotic Kinase Nek2: SAR and Structural Characterization

por Whelligan, Daniel K., Solanki, Savade, Taylor, Dawn, Thomson, Douglas W., Cheung, Kwai-Ming J., Boxall, Kathy, Mas-Droux, Corine, Barillari, Caterina, Burns, Samantha, Grummitt, Charles G., Collins, Ian, van Montfort, Rob L. M., Aherne, G. Wynne, Bayliss, Richard, Hoelder, Swen
Publicado 2010