An inter­molecular dative B←N bond in 5-(4,4,5,5-tetra­methyl-1,3,2-dioxa­borolan-2-yl)-1,3-thia­zole

por Sopková-de Oliveira Santos, Jana, Primas, Nicolas, Lohier, Jean-François, Bouillon, Alexandre, Rault, Sylvain
Publicado 2009

Computational Tool to Design Small Synthetic Inhibitors Selective for XIAP-BIR3 Domain

por Farag, Marc, Kieffer, Charline, Guedeney, Nicolas, Voisin-Chiret, Anne Sophie, Sopkova-de Oliveira Santos, Jana
Publicado 2023

tert-Butyl 6-bromo-1,4-dimethyl-9H-carbazole-9-carboxyl­ate

por Lohier, Jean-François, Caruso, Anna, Sopková-de Oliveira Santos, Jana, Lancelot, Jean-Charles, Rault, Sylvain
Publicado 2010

Development of Novel Potential Pleiotropic Compounds of Interest in Alzheimer’s Disease Treatment through Rigidification Strategy

por Lecoutey, Cédric, Legay, Rémi, Davis, Audrey, Sopková-de Oliveira Santos, Jana, Dallemagne, Patrick, Rochais, Christophe
Publicado 2021

Straightforward Access to a New Class of Dual DYRK1A/CLK1 Inhibitors Possessing a Simple Dihydroquinoline Core

por Ţînţaş, Mihaela-Liliana, Peauger, Ludovic, Alix, Florent, Papamicaël, Cyril, Besson, Thierry, Sopková-de Oliveira Santos, Jana, Gembus, Vincent, Levacher, Vincent
Publicado 2022

Rational design of novel benzisoxazole derivatives with acetylcholinesterase inhibitory and serotoninergic 5-HT(4) receptors activities for the treatment of Alzheimer’s disease

por Lalut, Julien, Payan, Hugo, Davis, Audrey, Lecoutey, Cédric, Legay, Rémi, Sopkova-de Oliveira Santos, Jana, Claeysen, Sylvie, Dallemagne, Patrick, Rochais, Christophe
Publicado 2020

First Synthesis of Racemic Trans Propargylamino-Donepezil, a Pleiotrope Agent Able to Both Inhibit AChE and MAO-B, with Potential Interest against Alzheimer’s Disease

por Guieu, Benjamin, Lecoutey, Cedric, Legay, Rémi, Davis, Audrey, Sopkova de Oliveira Santos, Jana, Altomare, Cosimo Damiano, Catto, Marco, Rochais, Christophe, Dallemagne, Patrick
Publicado 2020

Description of Joint Alterations Observed in a Family Carrying p.Asn453Ser COMP Variant: Clinical Phenotypes, In Silico Prediction of Functional Impact on COMP Protein and Stabilit...

por Rochoux, Quitterie, Sopkova-de Oliveira Santos, Jana, Marcelli, Christian, Rovelet-Lecrux, Anne, Chevallier, Virginie, Dutheil, Jean-Jacques, Leclercq, Sylvain, Boumédiene, Karim, Baugé, Catherine, Aury-Landas, Juliette
Publicado 2021

Inhibiting Acetylcholinesterase to Activate Pleiotropic Prodrugs with Therapeutic Interest in Alzheimer’s Disease

por Toublet, François-Xavier, Lecoutey, Cédric, Lalut, Julien, Hatat, Bérénice, Davis, Audrey, Since, Marc, Corvaisier, Sophie, Freret, Thomas, Sopkova de Oliveira Santos, Jana, Claeysen, Sylvie, Boulouard, Michel, Dallemagne, Patrick, Rochais, Christophe
Publicado 2019

Drug Repurposing: Deferasirox Inhibits the Anti-Apoptotic Activity of Mcl-1

por Bourafai-Aziez, Asma, Benabderrahmane, Mohammed, Paysant, Hippolyte, Weiswald, Louis-Bastien, Poulain, Laurent, Carlier, Ludovic, Ravault, Delphine, Jouanne, Marie, Coadou, Gaël, Oulyadi, Hassan, Voisin-Chiret, Anne-Sophie, Sopková-de Oliveira Santos, Jana, Sebban, Muriel
Publicado 2021

Discovery of Bis-Imidazoline Derivatives as New CXCR4 Ligands

por Zhou, Zhicheng, Staropoli, Isabelle, Brelot, Anne, Suzanne, Peggy, Lesnard, Aurélien, Fontaine, Fanny, Perato, Serge, Rault, Sylvain, Helynck, Olivier, Arenzana-Seisdedos, Fernando, Sopkova-de Oliveira Santos, Jana, Lagane, Bernard, Munier-Lehmann, Hélène, Colin, Philippe
Publicado 2023