Identification of Bichalcones as Sirtuin Inhibitors by Virtual Screening and In Vitro Testing

por Karaman, Berin, Alhalabi, Zayan, Swyter, Sören, Mihigo, Shetonde O., Andrae-Marobela, Kerstin, Jung, Manfred, Sippl, Wolfgang, Ntie-Kang, Fidele
Publicado 2018

Azologization and repurposing of a hetero-stilbene-based kinase inhibitor: towards the design of photoswitchable sirtuin inhibitors

por Grathwol, Christoph W, Wössner, Nathalie, Swyter, Sören, Smith, Adam C, Tapavicza, Enrico, Hofstetter, Robert K, Bodtke, Anja, Jung, Manfred, Link, Andreas
Publicado 2019

Sirtuin 1 Inhibiting Thiocyanates (S1th)—A New Class of Isotype Selective Inhibitors of NAD(+) Dependent Lysine Deacetylases

por Wössner, Nathalie, Alhalabi, Zayan, González, Jessica, Swyter, Sören, Gan, Jin, Schmidtkunz, Karin, Zhang, Lin, Vaquero, Alejandro, Ovaa, Huib, Einsle, Oliver, Sippl, Wolfgang, Jung, Manfred
Publicado 2020