Recent Advances in the Synthesis of Polyamine Derivatives and Their Applications

por Nichugovskiy, Artemiy, Tron, Gian Cesare, Maslov, Mikhail
Publicado 2021

Visible-Light Photoredox Catalysis in Water

por Russo, Camilla, Brunelli, Francesca, Tron, Gian Cesare, Giustiniano, Mariateresa
Publicado 2022

The Dark Side of Isocyanides: Visible-Light Photocatalytic Activity in the Oxidative Functionalization of C(sp(3))–H Bonds

por Russo, Camilla, Amato, Jussara, Tron, Gian Cesare, Giustiniano, Mariateresa
Publicado 2021

The 115 Years Old Multicomponent Bargellini Reaction: Perspectives and New Applications

por Serafini, Marta, Murgia, Ilaria, Giustiniano, Mariateresa, Pirali, Tracey, Tron, Gian Cesare
Publicado 2021

Icilio Guareschi and his amazing “1897 reaction”

por Tron, Gian Cesare, Minassi, Alberto, Sorba, Giovanni, Fausone, Mara, Appendino, Giovanni
Publicado 2021

Expanding the Chemical Space of Drug-like Passerini Compounds: Can α-Acyloxy Carboxamides Be Considered Hard Drugs?

por Brunelli, Francesca, Ceresa, Chiara, Fracchia, Letizia, Tron, Gian Cesare, Aprile, Silvio
Publicado 2022

Visible-Light Photocatalytic Functionalization of Isocyanides for the Synthesis of Secondary Amides and Ketene Aminals

por Cannalire, Rolando, Amato, Jussara, Summa, Vincenzo, Novellino, Ettore, Tron, Gian Cesare, Giustiniano, Mariateresa
Publicado 2020

Tritylamine as an Ammonia Surrogate in the Ugi Reaction Provides Access to Unprecedented 5-Sulfamido Oxazoles Using Burgess-type Reagents

por Bhela, Irene Preet, Serafini, Marta, Del Grosso, Erika, Tron, Gian Cesare, Pirali, Tracey
Publicado 2021

Data on metabolic stability, aqueous solubility and CYP inhibition of novel triazole-based nicotinamide phosphoribosyltransferase (NAMPT) inhibitors

por Aprile, Silvio, Galli, Ubaldina, Tron, Gian Cesare, Del Grosso, Erika, Travelli, Cristina, Grosa, Giorgio
Publicado 2019

What’s in a Name? Drug Nomenclature and Medicinal Chemistry Trends using INN Publications

por Serafini, Marta, Cargnin, Sarah, Massarotti, Alberto, Tron, Gian Cesare, Pirali, Tracey, Genazzani, Armando A.
Publicado 2021

Recent Advances in NAMPT Inhibitors: A Novel Immunotherapic Strategy

por Galli, Ubaldina, Colombo, Giorgia, Travelli, Cristina, Tron, Gian Cesare, Genazzani, Armando A., Grolla, Ambra A.
Publicado 2020

The Guareschi Pyridine Scaffold as a Valuable Platform for the Identification of Selective PI3K Inhibitors

por Galli, Ubaldina, Ciraolo, Elisa, Massarotti, Alberto, Margaria, Jean Piero, Sorba, Giovanni, Hirsch, Emilio, Tron, Gian Cesare
Publicado 2015

Photomicellar Catalyzed Synthesis of Amides from Isocyanides: Optimization, Scope, and NMR Studies of Photocatalyst/Surfactant Interactions

por Cannalire, Rolando, Santoro, Federica, Russo, Camilla, Graziani, Giulia, Tron, Gian Cesare, Carotenuto, Alfonso, Brancaccio, Diego, Giustiniano, Mariateresa
Publicado 2021

Exploiting the Nucleophilicity of the Nitrogen Atom of Imidazoles: One-Pot Three-Component Synthesis of Imidazo-Pyrazines

por Galli, Ubaldina, Hysenlika, Rejdia, Meneghetti, Fiorella, Del Grosso, Erika, Pelliccia, Sveva, Novellino, Ettore, Giustiniano, Mariateresa, Tron, Gian Cesare
Publicado 2019

The NAMPT inhibitor FK866 reverts the damage in spinal cord injury

por Esposito, Emanuela, Impellizzeri, Daniela, Mazzon, Emanuela, Fakhfouri, Gohar, Rahimian, Reza, Travelli, Cristina, Tron, Gian Cesare, Genazzani, Armando A, Cuzzocrea, Salvatore
Publicado 2012

Synthesis of Novel Lipophilic Polyamines via Ugi Reaction and Evaluation of Their Anticancer Activity

por Nichugovskiy, Artemiy, Maksimova, Varvara, Trapeznikova, Ekaterina, Eshtukova-Shcheglova, Elizaveta, Ivanov, Igor, Yakubovskaya, Marianna, Kirsanov, Kirill, Cheshkov, Dmitry, Tron, Gian Cesare, Maslov, Mikhail
Publicado 2022

Structure activity relationship studies on Amb639752: toward the identification of a common pharmacophoric structure for DGKα inhibitors

por Velnati, Suresh, Massarotti, Alberto, Antona, Annamaria, Talmon, Maria, Fresu, Luigia Grazia, Galetto, Alessandra Silvia, Capello, Daniela, Bertoni, Alessandra, Mercalli, Valentina, Graziani, Andrea, Tron, Gian Cesare, Baldanzi, Gianluca
Publicado 2019

Identification of a novel DGKα inhibitor for XLP-1 therapy by virtual screening

por Velnati, Suresh, Ruffo, Elisa, Massarotti, Alberto, Talmon, Maria, Varma, Konduru Sai Sandeep, Gesu, Alessandro, Fresu, Luigia Grazia, Snow, Andrew L., Bertoni, Alessandra, Capello, Daniela, Tron, Gian Cesare, Graziani, Andrea, Baldanzi, Gianluca
Publicado 2018

Synthesis and Characterization of Bis-Triazolyl-Pyridine Derivatives as Noncanonical DNA-Interacting Compounds

por Di Porzio, Anna, Galli, Ubaldina, Amato, Jussara, Zizza, Pasquale, Iachettini, Sara, Iaccarino, Nunzia, Marzano, Simona, Santoro, Federica, Brancaccio, Diego, Carotenuto, Alfonso, De Tito, Stefano, Biroccio, Annamaria, Pagano, Bruno, Tron, Gian Cesare, Randazzo, Antonio
Publicado 2021

Identification of a Potent Phosphoinositide 3‐Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs

por Pirali, Tracey, Ciraolo, Elisa, Aprile, Silvio, Massarotti, Alberto, Berndt, Alex, Griglio, Alessia, Serafini, Marta, Mercalli, Valentina, Landoni, Clarissa, Campa, Carlo Cosimo, Margaria, Jean Piero, Silva, Rangel L., Grosa, Giorgio, Sorba, Giovanni, Williams, Roger, Hirsch, Emilio, Tron, Gian Cesare
Publicado 2017