FKBP Ligands—Where We Are and Where to Go?

por Kolos, Jürgen M., Voll, Andreas M., Bauder, Michael, Hausch, Felix
Publicado 2018

Macrocyclic FKBP51 Ligands Define a Transient Binding Mode with Enhanced Selectivity

por Voll, Andreas M., Meyners, Christian, Taubert, Martha C., Bajaj, Thomas, Heymann, Tim, Merz, Stephanie, Charalampidou, Anna, Kolos, Jürgen, Purder, Patrick L., Geiger, Thomas M., Wessig, Pablo, Gassen, Nils C., Bracher, Andreas, Hausch, Felix
Publicado 2021

Picomolar FKBP inhibitors enabled by a single water-displacing methyl group in bicyclic [4.3.1] aza-amides

por Kolos, Jürgen M., Pomplun, Sebastian, Jung, Sascha, Rieß, Benedikt, Purder, Patrick L., Voll, Andreas M., Merz, Stephanie, Gnatzy, Monika, Geiger, Thomas M., Quist-Løkken, Ingrid, Jatzlau, Jerome, Knaus, Petra, Holien, Toril, Bracher, Andreas, Meyners, Christian, Czodrowski, Paul, Krewald, Vera, Hausch, Felix
Publicado 2021