(Hetero)aryl substituted thiazol-2,4-yl scaffold as human carbonic anhydrase I, II, VII and XIV activators

por Rami, Marouan, Winum, Jean-Yves, Supuran, Claudiu T., Melnyk, Patricia, Yous, Saïd
Publicado 2019

Carbazole scaffolds in cancer therapy: a review from 2012 to 2018

por Issa, Samar, Prandina, Anthony, Bedel, Nicolas, Rongved, Pål, Yous, Saïd, Le Borgne, Marc, Bouaziz, Zouhair
Publicado 2019

Novel Conformationally Constrained Analogues of Agomelatine as New Melatoninergic Ligands

por Rami, Marouan, Landagaray, Elodie, Ettaoussi, Mohamed, Boukhalfa, Koussayla, Caignard, Daniel-Henri, Delagrange, Philippe, Berthelot, Pascal, Yous, Saïd
Publicado 2012

Design, synthesis and evaluation of 2-aryl benzoxazoles as promising hit for the A(2A) receptor

por Duroux, Romain, Renault, Nicolas, Cuelho, Joana Esteves, Agouridas, Laurence, Blum, David, Lopes, Luisa V., Melnyk, Patricia, Yous, Saïd
Publicado 2017

Bitopic fluorescent antagonists of the A(2A) adenosine receptor based on pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine functionalized congeners

por Duroux, Romain, Ciancetta, Antonella, Mannes, Philip, Yu, Jinha, Boyapati, Shireesha, Gizewski, Elizabeth, Yous, Said, Ciruela, Francisco, Auchampach, John A., Gao, Zhan-Guo, Jacobson, Kenneth A.
Publicado 2017

New Radioligands for Describing the Molecular Pharmacology of MT(1) and MT(2) Melatonin Receptors

por Legros, Céline, Matthey, Ulrich, Grelak, Teresa, Pedragona-Moreau, Sandrine, Hassler, Werner, Yous, Saïd, Thomas, Emmanuel, Suzenet, Franck, Folleas, Benoît, Lefoulon, François, Berthelot, Pascal, Caignard, Daniel-Henri, Guillaumet, Gérald, Delagrange, Philippe, Brayer, Jean-Louis, Nosjean, Olivier, Boutin, Jean A.
Publicado 2013

XFEL structures of the human MT(2) melatonin receptor reveal basis of subtype selectivity

por Johansson, Linda C., Stauch, Benjamin, McCorvy, John D., Han, Gye Won, Patel, Nilkanth, Huang, Xi-Ping, Batyuk, Alexander, Gati, Cornelius, Slocum, Samuel T., Li, Chufeng, Grandner, Jessica M., Hao, Shuming, Olsen, Reid H.J., Tribo, Alexandra R., Zaare, Sahba, Zhu, Lan, Zatsepin, Nadia A., Weierstall, Uwe, Yous, Saïd, Stevens, Raymond C., Liu, Wei, Roth, Bryan L., Katritch, Vsevolod, Cherezov, Vadim
Publicado 2019

Structural basis for ligand recognition at the human MT(1) melatonin receptor

por Stauch, Benjamin, Johansson, Linda C., McCorvy, John D., Patel, Nilkanth, Han, Gye Won, Huang, Xi-Ping, Gati, Cornelius, Batyuk, Alexander, Slocum, Samuel T., Ishchenko, Andrii, Brehm, Wolfgang, White, Thomas A., Michaelian, Nairie, Madsen, Caleb, Zhu, Lan, Grant, Thomas D., Grandner, Jessica M., Shiriaeva, Anna, Olsen, Reid H.J., Tribo, Alexandra R., Yous, Saïd, Stevens, Raymond C., Weierstall, Uwe, Katritch, Vsevolod, Roth, Bryan L., Liu, Wei, Cherezov, Vadim
Publicado 2019