2-((1H-Benzo[d]imidazol-2-yl)amino)benzo[d]thiazole-6-sulphonamides: a class of carbonic anhydrase II and VII-selective inhibitors

por Abdoli, Morteza, Supuran, Claudiu T., Žalubovskis, Raivis
Publicado 2023

4-(3-Alkyl/benzyl-guanidino)benzenesulfonamides as selective carbonic anhydrase VII inhibitors

por Abdoli, Morteza, Giovannuzzi, Simone, Supuran, Claudiu T., Žalubovskis, Raivis
Publicado 2022

4-Cyanamidobenzenesulfonamide derivatives: a novel class of human and bacterial carbonic anhydrase inhibitors

por Abdoli, Morteza, Bonardi, Alessandro, Supuran, Claudiu T., Žalubovskis, Raivis
Publicado 2022

Investigation of novel alkyl/benzyl (4-sulphamoylphenyl)carbamimidothioates as carbonic anhydrase inhibitors

por Abdoli, Morteza, Bonardi, Alessandro, Supuran, Claudiu T., Žalubovskis, Raivis
Publicado 2023

3H-1,2-Benzoxaphosphepine 2-oxides as selective inhibitors of carbonic anhydrase IX and XII

por Pustenko, Aleksandrs, Balašova, Anastasija, Nocentini, Alessio, Supuran, Claudiu T., Žalubovskis, Raivis
Publicado 2022

1,2,3-Benzoxathiazine-2,2-dioxides – effective inhibitors of human carbonic anhydrases

por Ivanova, Jekaterina, Abdoli, Morteza, Nocentini, Alessio, Žalubovskis, Raivis, Supuran, Claudiu T.
Publicado 2022

Derivatives of 4-methyl-1,2,3-benzoxathiazine 2,2-dioxide as selective inhibitors of human carbonic anhydrases IX and XII over the cytosolic isoforms I and II

por Ivanova, Jekaterīna, Abdoli, Morteza, Nocentini, Alessio, Žalubovskis, Raivis, Supuran, Claudiu T.
Publicado 2023

Benzenesulfonamides Incorporating Hydantoin Moieties Effectively Inhibit Eukaryoticand Human Carbonic Anhydrases

por Abdoli, Morteza, De Luca, Viviana, Capasso, Clemente, Supuran, Claudiu T., Žalubovskis, Raivis
Publicado 2022

Novel thiazolone-benzenesulphonamide inhibitors of human and bacterial carbonic anhydrases

por Abdoli, Morteza, De Luca, Viviana, Capasso, Clemente, Supuran, Claudiu T., Žalubovskis, Raivis
Publicado 2023

Aryl derivatives of 3H-1,2-benzoxaphosphepine 2-oxides as inhibitors of cancer-related carbonic anhydrase isoforms IX and XII

por Balašova, Anastasija, Pustenko, Aleksandrs, Nocentini, Alessio, Vullo, Daniela, Supuran, Claudiu T., Žalubovskis, Raivis
Publicado 2023

May 1,2-Dithiolane-4-carboxylic Acid and Its Derivatives Serve as a Specific Thioredoxin Reductase 1 Inhibitor?

por Nikitjuka, Anna, Krims-Davis, Kristaps, Kaņepe-Lapsa, Iveta, Ozola, Melita, Žalubovskis, Raivis
Publicado 2023

Sulfocoumarins as dual inhibitors of human carbonic anhydrase isoforms IX/XII and of human thioredoxin reductase

por Krasavin, Mikhail, Žalubovskis, Raivis, Grandāne, Aiga, Domračeva, Ilona, Zhmurov, Petr, Supuran, Claudiu T.
Publicado 2020

7-Acylamino-3H-1,2-benzoxathiepine 2,2-dioxides as new isoform-selective carbonic anhydrase IX and XII inhibitors

por Pustenko, Aleksandrs, Nocentini, Alessio, Balašova, Anastasija, Krasavin, Mikhail, Žalubovskis, Raivis, Supuran, Claudiu T.
Publicado 2020

Aryl derivatives of 3H-1,2-benzoxathiepine 2,2-dioxide as carbonic anhydrase inhibitors

por Pustenko, Aleksandrs, Nocentini, Alessio, Balašova, Anastasija, Alafeefy, Ahmed, Krasavin, Mikhail, Žalubovskis, Raivis, Supuran, Claudiu T.
Publicado 2019

The antibiotic furagin and its derivatives are isoform-selective human carbonic anhydrase inhibitors

por Pustenko, Aleksandrs, Nocentini, Alessio, Gratteri, Paola, Bonardi, Alessandro, Vozny, Igor, Žalubovskis, Raivis, Supuran, Claudiu T.
Publicado 2020

Inhibition Studies on Human and Mycobacterial Carbonic Anhydrases with N-((4-Sulfamoylphenyl)carbamothioyl) Amides

por Abdoli, Morteza, Bonardi, Alessandro, Paoletti, Niccolò, Aspatwar, Ashok, Parkkila, Seppo, Gratteri, Paola, Supuran, Claudiu T., Žalubovskis, Raivis
Publicado 2023

3H-1,2-benzoxathiepine 2,2-dioxides: a new class of isoform-selective carbonic anhydrase inhibitors

por Pustenko, Aleksandrs, Stepanovs, Dmitrijs, Žalubovskis, Raivis, Vullo, Daniela, Kazaks, Andris, Leitans, Janis, Tars, Kaspars, Supuran, Claudiu T.
Publicado 2017

Combining carbonic anhydrase and thioredoxin reductase inhibitory motifs within a single molecule dramatically increases its cytotoxicity

por Krasavin, Mikhail, Sharonova, Tatiana, Sharoyko, Vladimir, Zhukovsky, Daniil, Kalinin, Stanislav, Žalubovskis, Raivis, Tennikova, Tatiana, Supuran, Claudiu T.
Publicado 2020

Design, synthesis, and biological evaluation of novel derivatives of dithiodiglycolic acid prepared via oxidative coupling of thiols

por Bakulina, Olga, Bannykh, Anton, Jovanović, Mirna, Domračeva, Ilona, Podolski-Renić, Ana, Žalubovskis, Raivis, Pešić, Milica, Dar’in, Dmitry, Krasavin, Mikhail
Publicado 2019

Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase

por Nocentini, Alessio, Angeli, Andrea, Carta, Fabrizio, Winum, Jean-Yves, Zalubovskis, Raivis, Carradori, Simone, Capasso, Clemente, Donald, William A., Supuran, Claudiu T.
Publicado 2021