Substituted N-Phenylpyrazine-2-carboxamides: Synthesis and Antimycobacterial Evaluation

por Doležal, Martin, Zitko, Jan, Kešetovičová, Diana, Kuneš, Jiří, Svobodová, Michaela
Publicado 2009

Towards Novel 3-Aminopyrazinamide-Based Prolyl-tRNA Synthetase Inhibitors: In Silico Modelling, Thermal Shift Assay and Structural Studies

por Pang, Luping, Weeks, Stephen D., Juhás, Martin, Strelkov, Sergei V., Zitko, Jan, Van Aerschot, Arthur
Publicado 2021

Synthesis, Biological Evaluation, and In Silico Modeling of N-Substituted Quinoxaline-2-Carboxamides

por Bouz, Ghada, Bouz, Sarah, Janďourek, Ondřej, Konečná, Klára, Bárta, Pavel, Vinšová, Jarmila, Doležal, Martin, Zitko, Jan
Publicado 2021

Design, Synthesis and Evaluation of N-pyrazinylbenzamides as Potential Antimycobacterial Agents

por Zitko, Jan, Mindlová, Alžběta, Valášek, Ondřej, Jand’ourek, Ondřej, Paterová, Pavla, Janoušek, Jiří, Konečná, Klára, Doležal, Martin
Publicado 2018

Synthesis of Novel Pyrazinamide Derivatives Based on 3-Chloropyrazine-2-carboxamide and Their Antimicrobial Evaluation

por Jandourek, Ondrej, Tauchman, Marek, Paterova, Pavla, Konecna, Klara, Navratilova, Lucie, Kubicek, Vladimir, Holas, Ondrej, Zitko, Jan, Dolezal, Martin
Publicado 2017

Synthesis, Antimycobacterial, Antifungal and Photosynthesis-Inhibiting Activity of Chlorinated N-phenylpyrazine-2-carboxamides †

por Dolezal, Martin, Zitko, Jan, Osicka, Zdenek, Kunes, Jiri, Vejsova, Marcela, Buchta, Vladimir, Dohnal, Jiri, Jampilek, Josef, Kralova, Katarina
Publicado 2010

New Potentially Active Pyrazinamide Derivatives Synthesized Under Microwave Conditions

por Jandourek, Ondrej, Dolezal, Martin, Kunes, Jiri, Kubicek, Vladimir, Paterova, Pavla, Pesko, Matus, Buchta, Vladimir, Kralova, Katarina, Zitko, Jan
Publicado 2014

Adenosine-Mimicking Derivatives of 3-Aminopyrazine-2-Carboxamide: Towards Inhibitors of Prolyl-tRNA Synthetase with Antimycobacterial Activity

por Pallabothula, Vinod Sukanth Kumar, Kerda, Marek, Juhás, Martin, Janďourek, Ondřej, Konečná, Klára, Bárta, Pavel, Paterová, Pavla, Zitko, Jan
Publicado 2022

5-Alkylamino-N-phenylpyrazine-2-carboxamides: Design, Preparation, and Antimycobacterial Evaluation

por Ambrożkiewicz, Weronika, Kučerová-Chlupáčová, Marta, Janďourek, Ondřej, Konečná, Klára, Paterová, Pavla, Bárta, Pavel, Vinšová, Jarmila, Doležal, Martin, Zitko, Jan
Publicado 2020

3-Substituted N-Benzylpyrazine-2-carboxamide Derivatives: Synthesis, Antimycobacterial and Antibacterial Evaluation

por Semelková, Lucia, Janďourek, Ondřej, Konečná, Klára, Paterová, Pavla, Navrátilová, Lucie, Trejtnar, František, Kubíček, Vladimír, Kuneš, Jiří, Doležal, Martin, Zitko, Jan
Publicado 2017

Synthesis, Antimycobacterial Activity and In Vitro Cytotoxicity of 5-Chloro-N-phenylpyrazine-2-carboxamides

por Zitko, Jan, Servusová, Barbora, Paterová, Pavla, Mandíková, Jana, Kubíček, Vladimír, Kučera, Radim, Hrabcová, Veronika, Kuneš, Jiří, Soukup, Ondřej, Doležal, Martin
Publicado 2013

Derivatives of 3-Aminopyrazine-2-carboxamides: Synthesis, Antimicrobial Evaluation, and in Vitro Cytotoxicity

por Bouz, Ghada, Semelková, Lucia, Janďourek, Ondřej, Konečná, Klára, Paterová, Pavla, Navrátilová, Lucie, Kubíček, Vladimír, Kuneš, Jiří, Doležal, Martin, Zitko, Jan
Publicado 2019

Ureidopyrazine Derivatives: Synthesis and Biological Evaluation as Anti-Infectives and Abiotic Elicitors

por Bouz, Ghada, Juhás, Martin, Niklová, Pavlína, Janďourek, Ondřej, Paterová, Pavla, Janoušek, Jiří, Tůmová, Lenka, Kovalíková, Zuzana, Kastner, Petr, Doležal, Martin, Zitko, Jan
Publicado 2017

Design, Synthesis, Antimycobacterial Evaluation, and In Silico Studies of 3-(Phenylcarbamoyl)-pyrazine-2-carboxylic Acids

por Semelková, Lucia, Janošcová, Petra, Fernandes, Carlos, Bouz, Ghada, Janďourek, Ondřej, Konečná, Klára, Paterová, Pavla, Navrátilová, Lucie, Kuneš, Jiří, Doležal, Martin, Zitko, Jan
Publicado 2017

Synthesis and Biological Evaluation of N-Alkyl-3-(alkylamino)-pyrazine-2-carboxamides

por Semelkova, Lucia, Konecna, Klara, Paterova, Pavla, Kubicek, Vladimir, Kunes, Jiri, Novakova, Lucie, Marek, Jan, Naesens, Lieve, Pesko, Matus, Kralova, Katarina, Dolezal, Martin, Zitko, Jan
Publicado 2015

Substituted N-(Pyrazin-2-yl)benzenesulfonamides; Synthesis, Anti-Infective Evaluation, Cytotoxicity, and In Silico Studies

por Bouz, Ghada, Juhás, Martin, Pausas Otero, Lluis, Paredes de la Red, Cristina, Janďourek, Ondřej, Konečná, Klára, Paterová, Pavla, Kubíček, Vladimír, Janoušek, Jiří, Doležal, Martin, Zitko, Jan
Publicado 2019

N-Pyrazinoyl Substituted Amino Acids as Potential Antimycobacterial Agents—the Synthesis and Biological Evaluation of Enantiomers

por Juhás, Martin, Kučerová, Lucie, Horáček, Ondřej, Janďourek, Ondřej, Kubíček, Vladimír, Konečná, Klára, Kučera, Radim, Bárta, Pavel, Janoušek, Jiří, Paterová, Pavla, Kuneš, Jiří, Doležal, Martin, Zitko, Jan
Publicado 2020

Correction: Juhás et al. Improving Antimicrobial Activity and Physico-Chemical Properties by Isosteric Replacement of 2-Aminothiazole with 2-Aminooxazole. Pharmaceuticals 2022, 15,...

por Juhás, Martin, Bachtíková, Andrea, Nawrot, Daria Elżbieta, Hatoková, Paulína, Pallabothula, Vinod Sukanth Kumar, Diepoltová, Adéla, Janďourek, Ondřej, Bárta, Pavel, Konečná, Klára, Paterová, Pavla, Šesták, Vít, Zitko, Jan
Publicado 2023

Improving Antimicrobial Activity and Physico-Chemical Properties by Isosteric Replacement of 2-Aminothiazole with 2-Aminooxazole

por Juhás, Martin, Bachtíková, Andrea, Nawrot, Daria Elżbieta, Hatoková, Paulína, Pallabothula, Vinod Sukanth Kumar, Diepoltová, Adéla, Janďourek, Ondřej, Bárta, Pavel, Konečná, Klára, Paterová, Pavla, Šesták, Vít, Zitko, Jan
Publicado 2022

The Forty-Sixth Euro Congress on Drug Synthesis and Analysis: Snapshot †

por Mucaji, Pavel, Atanasov, Atanas G., Bak, Andrzej, Kozik, Violetta, Sieron, Karolina, Olsen, Mark, Pan, Weidong, Liu, Yazhou, Hu, Shengchao, Lan, Junjie, Haider, Norbert, Musiol, Robert, Vanco, Jan, Diederich, Marc, Ji, Seungwon, Zitko, Jan, Wang, Dongdong, Agbaba, Danica, Nikolic, Katarina, Oljacic, Slavica, Vucicevic, Jelica, Jezova, Daniela, Tsantili-Kakoulidou, Anna, Tsopelas, Fotios, Giaginis, Constantinos, Kowalska, Teresa, Sajewicz, Mieczyslaw, Silberring, Jerzy, Mielczarek, Przemyslaw, Smoluch, Marek, Jendrzejewska, Izabela, Polanski, Jaroslaw, Jampilek, Josef
Publicado 2017