A Fluorescence‐Based Assay for Screening β‐Lactams Targeting the Mycobacterium tuberculosis Transpeptidase Ldt(Mt2)

por de Munnik, Mariska, Lohans, Christopher T., Langley, Gareth W., Bon, Corentin, Brem, Jürgen, Schofield, Christopher J.
Publicado 2019

αβ,α′β′-Diepoxyketones are mechanism-based inhibitors of nucleophilic cysteine enzymes

por de Munnik, Mariska, Lithgow, Jasper, Brewitz, Lennart, Christensen, Kirsten E., Bates, Robert H., Rodriguez-Miquel, Beatriz, Schofield, Christopher J.
Publicado 2023

Targeting the Mycobacterium tuberculosis transpeptidase Ldt(Mt2) with cysteine-reactive inhibitors including ebselen

por de Munnik, Mariska, Lohans, Christopher T., Lang, Pauline A., Langley, Gareth W., Malla, Tika R., Tumber, Anthony, Schofield, Christopher J., Brem, Jürgen
Publicado 2019

High-throughput screen with the l,d-transpeptidase Ldt(Mt2) of Mycobacterium tuberculosis reveals novel classes of covalently reacting inhibitors

por de Munnik, Mariska, Lang, Pauline A., De Dios Anton, Francisco, Cacho, Mónica, Bates, Robert H., Brem, Jürgen, Rodríguez Miquel, Beatriz, Schofield, Christopher J.
Publicado 2023

Non‐Hydrolytic β‐Lactam Antibiotic Fragmentation by l,d‐Transpeptidases and Serine β‐Lactamase Cysteine Variants

por Lohans, Christopher T., Chan, H. T. Henry, Malla, Tika R., Kumar, Kiran, Kamps, Jos J. A. G., McArdle, Darius J. B., van Groesen, Emma, de Munnik, Mariska, Tooke, Catherine L., Spencer, James, Paton, Robert S., Brem, Jürgen, Schofield, Christopher J.
Publicado 2019