A Straightforward Diphenylmethyl Protection Method and Deprotection of Some Pyrimidine Nucleosides

por Saudi, Milind, van Aerschot, Arthur
Publicado 2013

Using Chemical Approaches to Understand RNA Structure and Function in Biology

por Stetsenko, Dmitry A., van Aerschot, Arthur
Publicado 2012

Aminoacyl-tRNA Synthetases as Valuable Targets for Antimicrobial Drug Discovery

por Pang, Luping, Weeks, Stephen D., Van Aerschot, Arthur
Publicado 2021

Synthesis and evaluation of imidazole-4,5- and pyrazine-2,3-dicarboxamides targeting dengue and yellow fever virus()

por Saudi, Milind, Zmurko, Joanna, Kaptein, Suzanne, Rozenski, Jef, Neyts, Johan, Van Aerschot, Arthur
Publicado 2014

Hybridisation Potential of 1',3'-Di-O-methylaltropyranoside Nucleic Acids

por Venkatesham, Akkaladevi, Kachare, Dhuldeo, Schepers, Guy, Rozenski, Jef, Froeyen, Mathy, Van Aerschot, Arthur
Publicado 2015

Inhibition of MDR1 expression with altritol-modified siRNAs

por Fisher, Michael, Abramov, Mikhail, Van Aerschot, Arthur, Xu, Dong, Juliano, Rudolph L., Herdewijn, Piet
Publicado 2007

Propargylated Purine Deoxynucleosides: New Tools for Fluorescence Imaging Strategies

por Venkatesham, Akkaladevi, Pillalamarri, Sambasiva Rao, De Wit, Flore, Lescrinier, Eveline, Debyser, Zeger, Van Aerschot, Arthur
Publicado 2019

Towards Novel 3-Aminopyrazinamide-Based Prolyl-tRNA Synthetase Inhibitors: In Silico Modelling, Thermal Shift Assay and Structural Studies

por Pang, Luping, Weeks, Stephen D., Juhás, Martin, Strelkov, Sergei V., Zitko, Jan, Van Aerschot, Arthur
Publicado 2021

Partitioning of the initial catalytic steps of leucyl-tRNA synthetase is driven by an active site peptide-plane flip

por Pang, Luping, Zanki, Vladimir, Strelkov, Sergei V., Van Aerschot, Arthur, Gruic-Sovulj, Ita, Weeks, Stephen D.
Publicado 2022

A Trojan-Horse Peptide-Carboxymethyl-Cytidine Antibiotic from Bacillus amyloliquefaciens

por Serebryakova, Marina, Tsibulskaya, Darya, Mokina, Olga, Kulikovsky, Alexey, Nautiyal, Manesh, Van Aerschot, Arthur, Severinov, Konstantin, Dubiley, Svetlana
Publicado 2016

N-Alkylated Aminoacyl sulfamoyladenosines as Potential Inhibitors of Aminoacylation Reactions and Microcin C Analogues Containing D-Amino Acids

por Vondenhoff, Gaston H., Pugach, Ksenia, Gadakh, Bharat, Carlier, Laurence, Rozenski, Jef, Froeyen, Mathy, Severinov, Konstantin, Van Aerschot, Arthur
Publicado 2013

Synthesis and Biological Evaluation of Lipophilic Nucleoside Analogues as Inhibitors of Aminoacyl-tRNA Synthetases

por Nautiyal, Manesh, Gadakh, Bharat, De Graef, Steff, Pang, Luping, Khan, Masroor, Xun, Yi, Rozenski, Jef, Van Aerschot, Arthur
Publicado 2019

Synthetic strategy and antiviral evaluation of diamide containing heterocycles targeting dengue and yellow fever virus()

por Saudi, Milind, Zmurko, Joanna, Kaptein, Suzanne, Rozenski, Jef, Gadakh, Bharat, Chaltin, Patrick, Marchand, Arnaud, Neyts, Johan, Van Aerschot, Arthur
Publicado 2016

Structural Basis of Cysteine Ligase MshC Inhibition by Cysteinyl-Sulfonamides

por Pang, Luping, Lenders, Stijn, Osipov, Evgenii M., Weeks, Stephen D., Rozenski, Jef, Piller, Tatiana, Cappoen, Davie, Strelkov, Sergei V., Van Aerschot, Arthur
Publicado 2022

Synthesis and Biological Evaluation of 1,3-Dideazapurine-Like 7-Amino-5-Hydroxymethyl-Benzimidazole Ribonucleoside Analogues as Aminoacyl-tRNA Synthetase Inhibitors

por Zhang, Baole, Pang, Luping, Nautiyal, Manesh, De Graef, Steff, Gadakh, Bharat, Lescrinier, Eveline, Rozenski, Jef, Strelkov, Sergei V., Weeks, Stephen D., Van Aerschot, Arthur
Publicado 2020

Discovery of novel druggable pockets on polyomavirus VP1 through crystallographic fragment-based screening to develop capsid assembly inhibitors

por Osipov, Evgenii M., Munawar, Ali H., Beelen, Steven, Fearon, Daren, Douangamath, Alice, Wild, Conor, Weeks, Stephen D., Van Aerschot, Arthur, von Delft, Frank, Strelkov, Sergei V.
Publicado 2022

A large-scale chemical modification screen identifies design rules to generate siRNAs with high activity, high stability and low toxicity

por Bramsen, Jesper B., Laursen, Maria B., Nielsen, Anne F., Hansen, Thomas B., Bus, Claus, Langkjær, Niels, Babu, B. Ravindra, Højland, Torben, Abramov, Mikhail, Van Aerschot, Arthur, Odadzic, Dalibor, Smicius, Romualdas, Haas, Jens, Andree, Cordula, Barman, Jharna, Wenska, Malgorzata, Srivastava, Puneet, Zhou, Chuanzheng, Honcharenko, Dmytro, Hess, Simone, Müller, Elke, Bobkov, Georgii V., Mikhailov, Sergey N., Fava, Eugenio, Meyer, Thomas F., Chattopadhyaya, Jyoti, Zerial, Marino, Engels, Joachim W., Herdewijn, Piet, Wengel, Jesper, Kjems, Jørgen
Publicado 2009