Cargando…

Synthesis, In Silico Analysis, and Larvicidal Activity of New Bis-oxadiazole Derivatives

Twelve new 2,2′-bi(1,2,4-oxadiazole) derivatives containing heterocyclic and long-chain substituents have been synthesized by the condensation of aldehyde azines and oximes. In silico studies of these compounds revealed their good drug likeness and drug score. Some of the synthesized compounds show...

Descripción completa

Detalles Bibliográficos
Autores principales:	Balije, Rakesh, A, Prasad, Shyam, Perugu, Velidandi, Amar nath
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Pleiades Publishing 2023
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10036162/ http://dx.doi.org/10.1134/S1070428023010177

Ejemplares similares

Synthesis and Larvicidal Activity of Novel Thenoylhydrazide Derivatives
por: Song, Gao-Peng, et al.
Publicado: (2016)

Synthesis of Some Oxadiazole Derivatives as New Anticandidal Agents
por: Kaplancikli, Zafer Asim
Publicado: (2011)

Synthesis and Pharmacological Characterization of Metronidazole-Oxadiazole Derivatives
por: Mohammed, Mohsin, et al.
Publicado: (2023)

Synthesis and Antimicrobial Evaluation of Some New Oxadiazoles Derived from Phenylpropionohydrazides
por: Fuloria, Neeraj Kumar, et al.
Publicado: (2009)

Synthesis and Anticancer Evaluation of New 1,3,4-Oxadiazole Derivatives
por: Stecoza, Camelia Elena, et al.
Publicado: (2021)

A New Class of Glucosyl Thioureas: Synthesis and Larvicidal Activities
por: Wang, Ping-An, et al.
Publicado: (2016)

Synthesis, Characterization, and Biologic Activity of New Acyl Hydrazides and 1,3,4-Oxadiazole Derivatives
por: Zarafu, Irina, et al.
Publicado: (2020)

Biological activity of oxadiazole and thiadiazole derivatives
por: Atmaram, Upare Abhay, et al.
Publicado: (2022)

Antioxidant, Antimicrobial, Cytotoxicity, and Larvicidal Activities of Selected Synthetic Bis-Chalcones
por: Kuttithodi, Aswathi Moothakoottil, et al.
Publicado: (2022)

Design, Synthesis, In Silico and In Vitro Studies for New Nitric Oxide-Releasing Indomethacin Derivatives with 1,3,4-Oxadiazole-2-thiol Scaffold
por: Sava, Alexandru, et al.
Publicado: (2021)

Synthesis, Larvicidal Activities and Antifungal Activities of Novel Chlorantraniliprole Derivatives and Their Target in the Ryanodine Receptor
por: Chen, Qichao, et al.
Publicado: (2015)

1,3,4-Oxadiazole Derivatives: Synthesis, Characterization, Antimicrobial Potential, and Computational Studies
por: Bala, Suman, et al.
Publicado: (2014)

Design, synthesis, and biological activity of novel 1,2,4-oxadiazole derivatives
por: Zhu, Lingzhi, et al.
Publicado: (2020)

Synthesis of Oxadiazole-Thiadiazole Hybrids and Their Anticandidal Activity
por: Levent, Serkan, et al.
Publicado: (2017)

Synthesis and Bioassay of a New Class of Furanyl-1,3,4-Oxadiazole Derivatives
por: El Sadek, Mohamed M., et al.
Publicado: (2013)

Phytochemical Investigation of Three Cystoseira Species and Their Larvicidal Activity Supported with In Silico Studies
por: Aly, Shaza H., et al.
Publicado: (2023)

New 1,2,4-Oxadiazole Nortopsentin Derivatives with Cytotoxic Activity
por: Cascioferro, Stella, et al.
Publicado: (2019)

Simple and Efficient Synthesis of Diamino Derivatives of bis-1,2,4-oxadiazole via Tandem Staudinger/aza-Wittig Reaction
por: Xie, Hai, et al.
Publicado: (2023)

Synthesis, crystal structure and larvicidal activity of novel diamide derivatives against Culex pipiens
por: Wu, Rui, et al.
Publicado: (2012)

Evaluation of Antidiabetic Activity of Oxadiazole Derivative in Rats
por: Qazi, Adil Iqbal, et al.
Publicado: (2023)

Combined in Vitro and in Silico Studies for the Anticholinesterase Activity and Pharmacokinetics of Coumarinyl Thiazoles and Oxadiazoles
por: Ibrar, Aliya, et al.
Publicado: (2018)

A New and Efficient Method for the Synthesis of Novel 3-Acetyl Coumarins Oxadiazoles Derivatives with Expected Biological Activity
por: Sulaiman Al-Ayed, Abdullah, et al.
Publicado: (2014)

Synthesis of new 2-amino-1,3,4-oxadiazole derivatives with anti-salmonella typhi activity evaluation
por: Salama, Eid E.
Publicado: (2020)

Investigation of Novel Benzoxazole-Oxadiazole Derivatives as Effective Anti-Alzheimer’s Agents: In Vitro and In Silico Approaches
por: Anwar, Saeed, et al.
Publicado: (2023)

Synthesis, In Silico, and In Vitro Evaluation of Anti-Leishmanial Activity of Oxadiazoles and Indolizine Containing Compounds Flagged against Anti-Targets
por: Stevanovic, Strahinja, et al.
Publicado: (2019)

Synthesis and antifungal activities of novel nicotinamide derivatives containing 1,3,4-oxadiazole
por: Wu, Jian, et al.
Publicado: (2013)

Synthesis, Characterization and Anti-Inflammatory Activity of Some 1, 3,4 -Oxadiazole Derivatives
por: Kumar Singh, Arvind, et al.
Publicado: (2013)

Synthesis of novel oxadiazole derivatives and their cytotoxic activity against various cancer cell lines
por: SUCU, Bilgesu Onur, et al.
Publicado: (2022)

Synthesis and Chemometrics of Thymol and Carvacrol Derivatives as Larvicides against Aedes aegypti
por: Silva, Viviane Barros, et al.
Publicado: (2017)

Design, Synthesis, In Vivo, and In Silico Evaluation of Benzothiazoles Bearing a 1,3,4-Oxadiazole Moiety as New Antiepileptic Agents
por: Chauhan, Bharti, et al.
Publicado: (2023)

Design, Synthesis and Evaluation of New Bioactive Oxadiazole Derivatives as Anticancer Agents Targeting Bcl-2
por: Hamdy, Rania, et al.
Publicado: (2020)

Research progress on the synthesis and pharmacology of 1,3,4-oxadiazole and 1,2,4-oxadiazole derivatives: a mini review
por: Wang, Jing-Jing, et al.
Publicado: (2022)

Synthesis and Larvicidal Activity against Culex pipiens pallens of New Triazole Derivatives of Phrymarolin from Phryma leptostachya L.
por: Zhang, Ji-Wen, et al.
Publicado: (2013)

Synthesis of Oxadiazoles, Thiadiazoles and Triazoles Derived from Benzo[b]thiophene.
por: Sharba, A. Hussain K., et al.
Publicado: (2005)

Synthesis, Molecular Properties Prediction, and Anti-staphylococcal Activity of N-Acylhydrazones and New 1,3,4-Oxadiazole Derivatives
por: de Oliveira, Cledualdo Soares, et al.
Publicado: (2012)

Synthesis of new oxadiazol-phthalazinone derivatives with anti-proliferative activity; molecular docking, pro-apoptotic, and enzyme inhibition profile
por: Hekal, Mohamed H., et al.
Publicado: (2020)

Synthesis, characterization, molecular docking, and anticancer activities of new 1,3,4-oxadiazole-5-fluorocytosine hybrid derivatives
por: El Mansouri, Az-eddine, et al.
Publicado: (2022)

Anti-proliferative activity and characterization data on oxadiazole derivatives
por: Dukanya, et al.
Publicado: (2020)

Antimicrobial Activity of 1,3,4-Oxadiazole Derivatives
por: Glomb, Teresa, et al.
Publicado: (2021)

2,5-Bis(2,2,2-trifluoroethoxy)phenyl-tethered 1,3,4-Oxadiazoles Derivatives: Synthesis, In Silico Studies, and Biological Assessment as Potential Candidates for Anti-Cancer and Anti-Diabetic Agent
por: Shankara, Sathyanarayana D., et al.
Publicado: (2022)

Cannot write session to /tmp/vufind_sessions/sess_ghrdo904l6bjn1dvnvlhlb8021