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Synthesis and Biological Evaluation of Coumarin Triazoles as Dual Inhibitors of Cholinesterases and β-Secretase

[Image: see text] Coumarin is a naturally occurring bioactive pharmacophore with wide occurrence among central nervous system (CNS)-active small molecules. 8-Acetylcoumarin, one of the natural coumarins, is a mild inhibitor of cholinesterases and β-secretase, which are vital targets of Alzheimer’s d...

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Detalles Bibliográficos
Autores principales:	Sharma, Ankita, Bharate, Sandip B.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2023
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10061512/ https://www.ncbi.nlm.nih.gov/pubmed/37008108 http://dx.doi.org/10.1021/acsomega.2c07993

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