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Antiseizure Properties of Histamine H(3) Receptor Antagonists Belonging 3,4-Dihydroquinolin-2(1H)-Ones
H(3)R is becoming an attractive and promising target for epilepsy treatment as well as the discovery of antiepileptics. In this work, a series of 6-aminoalkoxy-3,4-dihydroquinolin-2(1H)-ones was prepared to screen their H(3)R antagonistic activities and antiseizure effects. The majority of the targe...
Autores principales: | Hua, Yi, Song, Mingxia, Guo, Qiaoyue, Luo, Yiqin, Deng, Xianqing, Huang, Yushan |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2023
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10144301/ https://www.ncbi.nlm.nih.gov/pubmed/37110645 http://dx.doi.org/10.3390/molecules28083408 |
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