Syntheses of 2- and 3-Substituted Morpholine Congeners via Ring Opening of 2-Tosyl-1,2-Oxazetidine

[Image: see text] Diastereoselective and diastereoconvergent syntheses of 2- and 3-substituted morpholine congeners are reported. Starting from tosyl-oxazatedine 1 and α-formyl carboxylates 2, base catalysis is utilized to yield morpholine hemiaminals. Their further synthetic elaborations allowed th...

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Detalles Bibliográficos
Autores principales: Kőnig, Bálint, Sztanó, Gábor, Holczbauer, Tamás, Soós, Tibor
Formato: Online Artículo Texto
Lenguaje:English
Publicado: American Chemical Society 2023
Acceso en línea:https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10167689/
https://www.ncbi.nlm.nih.gov/pubmed/37125664
http://dx.doi.org/10.1021/acs.joc.3c00207

Internet

https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10167689/
https://www.ncbi.nlm.nih.gov/pubmed/37125664
http://dx.doi.org/10.1021/acs.joc.3c00207

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