Cargando…

Design, synthesis, anticancer evaluation and molecular docking studies of 1,2,3-triazole incorporated 1,3,4-oxadiazole-Triazine derivatives

A new library of 1,2,3-triazole-incorporated 1,3,4-oxadiazole-triazine derivatives (9a-j) was designed, synthesized, and tested in vitro for anticancer activity against PC3 and DU-145 (prostate cancer), A549 (lung cancer), and MCF-7 (breast cancer) cancer cell lines using the MTT assay with etoposid...

Descripción completa

Detalles Bibliográficos
Autores principales:	Oggu, Sujana, Akshinthala, Parameswari, Katari, Naresh Kumar, Nagarapu, Laxmi Kumari, Malempati, Srimannarayana, Gundla, Rambabu, Jonnalagadda, Sreekantha Babu
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Elsevier 2023
Materias:	Research Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10189396/ https://www.ncbi.nlm.nih.gov/pubmed/37206039 http://dx.doi.org/10.1016/j.heliyon.2023.e15935

Ejemplares similares

New oxindole carboxamides as inhibitors of DENV NS5 RdRp: Design, synthesis, docking and Biochemical characterization
por: Koraboina, Chandra Prakash, et al.
Publicado: (2023)

Unique Quality by Design Approach for Developing HPLC and LC-MS Method for Estimation of Process and Degradation Impurities in Pibrentasvir, Antiviral Agent for Hepatitis C
por: Vemuri, Divya Kumar, et al.
Publicado: (2022)

Molecular Hybrids of Pyazolo[3,4-b]pyridine and Triazole: Design, Synthesis and In Vitro Antibacterial Studies
por: Bandaru, Narasimha Rao, et al.
Publicado: (2022)

Convenient synthesis, characterization and biological evaluation of novel 1-phenylcyclopropane carboxamide derivatives
por: Mahesh, Panasa, et al.
Publicado: (2023)

Antiproliferative Activity of New Pyrazole-4-sulfonamide Derivatives: Synthesis and Biological Evaluation
por: Mahesh, Panasa, et al.
Publicado: (2023)

Synthesis and Biological Evaluation of 1,2,3-Triazole Tethered Thymol-1,3,4-Oxadiazole Derivatives as Anticancer and Antimicrobial Agents
por: Almalki, Abdulraheem S. A., et al.
Publicado: (2021)

α-Glucosidase and α-Amylase Inhibitory Potentials of Quinoline–1,3,4-oxadiazole Conjugates Bearing 1,2,3-Triazole with Antioxidant Activity, Kinetic Studies, and Computational Validation
por: Cele, Nosipho, et al.
Publicado: (2022)

Synthesis of some new pyrazolo[1,5-a]pyrimidine, pyrazolo[5,1-c]triazine, 1,3,4-thiadiazole and pyridine derivatives containing 1,2,3-triazole moiety
por: Abdelriheem, Nadia A., et al.
Publicado: (2017)

Antimicrobial Activity of 1,3,4-Oxadiazole Derivatives
por: Glomb, Teresa, et al.
Publicado: (2021)

Synthesis, analgesic and anti-inflammatory activities of new methyl-imidazolyl-1,3,4-oxadiazoles and 1,2,4-triazoles
por: Almasirad, Ali, et al.
Publicado: (2014)

Synthesis of new, highly luminescent bis(2,2’-bithiophen-5-yl) substituted 1,3,4-oxadiazole, 1,3,4-thiadiazole and 1,2,4-triazole
por: Kostyuchenko, Anastasia S, et al.
Publicado: (2014)

1,2,3-Triazoles
por: Rachwal, S., et al.
Publicado: (2008)

Synthesis of Novel 2,5-Disubstituted-1,3,4-thiadiazoles Clubbed 1,2,4-Triazole, 1,3,4-Thiadiazole, 1,3,4-Oxadiazole and/or Schiff Base as Potential Antimicrobial and Antiproliferative Agents
por: Rezki, Nadjet, et al.
Publicado: (2015)

Synthesis of Biologically Relevant 1,2,3- and 1,3,4-Triazoles: From Classical Pathway to Green Chemistry
por: Gonnet, Lori, et al.
Publicado: (2021)

2-(1,2,4-triazole-5-yl)-1,3,4-oxadiazole as a novel building block for energetic materials
por: Dong, Zheting, et al.
Publicado: (2022)

5-Phenyl-1,3,4-oxadiazol-2-amine
por: Song, Man-Man, et al.
Publicado: (2012)

Anti-Cancer Activity of Derivatives of 1,3,4-Oxadiazole
por: Glomb, Teresa, et al.
Publicado: (2018)

1,3,4-Oxadiazoles by Ugi-Tetrazole and Huisgen Reaction
por: Wang, Qian, et al.
Publicado: (2019)

(1-(4-(5-Phenyl-1,3,4-oxadiazol-2-yl)phenyl)-1H-1,2,3-triazol-4-yl)-methylenyls α,ω-Bisfunctionalized 3- and 4-PEG: Synthesis and Photophysical Studies
por: Mohammed, Mohammed S., et al.
Publicado: (2023)

Cycloadditions of Noncomplementary Substituted 1,2,3-Triazines
por: Anderson, Erin D., et al.
Publicado: (2014)

Synthesis of Some New 1,3,4-Thiadiazole, Thiazole and Pyridine Derivatives Containing 1,2,3-Triazole Moiety
por: Abdelriheem, Nadia A., et al.
Publicado: (2017)

Electrophilic activation of nitroalkanes in efficient synthesis of 1,3,4-oxadiazoles
por: Aksenov, Alexander V., et al.
Publicado: (2019)

Synthesis and Anticancer Evaluation of New 1,3,4-Oxadiazole Derivatives
por: Stecoza, Camelia Elena, et al.
Publicado: (2021)

Green Chromatographic Method for Determination of Active Pharmaceutical Ingredient, Preservative, and Antioxidant in an Injectable Formulation: Robustness by Design Expert
por: Kowtharapu, Leela Prasad, et al.
Publicado: (2022)

2-[3,4-Dibutoxy-5-(5-phenyl-1,3,4-oxadiazol-2-yl)-2-thienyl]-5-phenyl-1,3,4-oxadiazole
por: Li, Hai-lin, et al.
Publicado: (2008)

2-Phenyl-5-(p-tolyl)-1,3,4-oxadiazole
por: Cordes, David B., et al.
Publicado: (2011)

Synthesis, Characterization and Biological Activity Studies of 1,3,4-Oxadiazole Analogs
por: Bhat, KI, et al.
Publicado: (2011)

Trifluoromethylpyridine 1,3,4-Oxadiazole Derivatives: Emerging Scaffolds as Bacterial Agents
por: Yu, Gang, et al.
Publicado: (2021)

Synthesis and Antimicrobial Activity of New 5-(2-Thienyl)-1,2,4-triazoles and 5-(2-Thienyl)-1,3,4-oxadiazoles and Related Derivatives
por: Al-Omar, Mohamed A.
Publicado: (2010)

Synthesis, Thermal, and Optical Properties of Tris(5‐aryl‐1,3,4‐oxadiazol‐2‐yl)‐1,3,5‐triazines, New Star‐Shaped Fluorescent Discotic Liquid Crystals
por: Tober, Natalie, et al.
Publicado: (2019)

Research progress on the synthesis and pharmacology of 1,3,4-oxadiazole and 1,2,4-oxadiazole derivatives: a mini review
por: Wang, Jing-Jing, et al.
Publicado: (2022)

Nanostructured Samarium Doped Fluorapatites and Their Catalytic Activity towards Synthesis of 1,2,4-Triazoles
por: Gangu, Kranthi Kumar, et al.
Publicado: (2016)

A comparison between observed and DFT calculations on structure of 5-(4-chlorophenyl)-2-amino-1,3,4-thiadiazole
por: Kerru, Nagaraju, et al.
Publicado: (2019)

Synthesis, Antimicrobial and Antiinflammatory Activity of 2,5-Disubstituted-1,3,4-oxadiazoles
por: Nagalakshmi, G.
Publicado: (2008)

5-(4-Methylphenyl)-1,3,4-oxadiazol-2-amine
por: Zheng, Juan, et al.
Publicado: (2012)

2,6-Dimethyl-4-(1,3,4-oxadiazol-2-yl)quinoline
por: Kashaev, Artyom G., et al.
Publicado: (2010)

Synthesis and Biological Evaluation of β-Aroylpropionic acid based 1,3,4-Oxadiazoles
por: Husain, A., et al.
Publicado: (2009)

Synthesis and antifungal activities of novel nicotinamide derivatives containing 1,3,4-oxadiazole
por: Wu, Jian, et al.
Publicado: (2013)

1,3,4-Oxadiazole Derivatives: Synthesis, Characterization, Antimicrobial Potential, and Computational Studies
por: Bala, Suman, et al.
Publicado: (2014)

Novel 2,5-disubstituted-1,3,4-oxadiazoles as anti-inflammatory drugs
por: Durgashivaprasad, Ega, et al.
Publicado: (2014)

Cannot write session to /tmp/vufind_sessions/sess_8euu26mslvfivtsm3rg4dqoc54