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Synthesis, Fluorine-18 Radiolabeling, and In Vivo PET Imaging of a Hydrophilic Fluorosulfotetrazine

The development of (18)F-fluorotetrazines, suitable for the radiolabeling of biologics such as proteins and antibodies by IEDDA ligation, represents a major challenge, especially for pre-targeting applications. The hydrophilicity of the tetrazine has clearly become a crucial parameter for the perfor...

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Detalles Bibliográficos
Autores principales:	Beaufrez, Jason, Guillouet, Stéphane, Seimbille, Yann, Perrio, Cécile
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2023
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10221973/ https://www.ncbi.nlm.nih.gov/pubmed/37242419 http://dx.doi.org/10.3390/ph16050636

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