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Inhibition Studies on Human and Mycobacterial Carbonic Anhydrases with N-((4-Sulfamoylphenyl)carbamothioyl) Amides

A library of structurally diverse N-((4-sulfamoylphenyl)carbamothioyl) amides was synthesized by selective acylation of easily accessible 4-thioureidobenzenesulfonamide with various aliphatic, benzylic, vinylic and aromatic acyl chlorides under mild conditions. Inhibition of three α-class cytosolic...

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Detalles Bibliográficos
Autores principales:	Abdoli, Morteza, Bonardi, Alessandro, Paoletti, Niccolò, Aspatwar, Ashok, Parkkila, Seppo, Gratteri, Paola, Supuran, Claudiu T., Žalubovskis, Raivis
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2023
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10222120/ https://www.ncbi.nlm.nih.gov/pubmed/37241761 http://dx.doi.org/10.3390/molecules28104020

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