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Synthesis of imidazo[1,2-a]pyridine-containing peptidomimetics by tandem of Groebke–Blackburn–Bienaymé and Ugi reactions

Peptidomimetics with a substituted imidazo[1,2-a]pyridine fragment were synthesized by a tandem of Groebke–Blackburn–Bienaymé and Ugi reactions. The target products contain substituted imidazo[1,2-a]pyridine and peptidomimetic moieties as pharmacophores with four diversity points introduced from rea...

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Detalles Bibliográficos
Autores principales:	Kolomiiets, Oleksandr V, Tsygankov, Alexander V, Kornet, Maryna N, Brazhko, Aleksander A, Musatov, Vladimir I, Chebanov, Valentyn A
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	Beilstein-Institut 2023
Materias:	Full Research Paper
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10241102/ https://www.ncbi.nlm.nih.gov/pubmed/37284590 http://dx.doi.org/10.3762/bjoc.19.53

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