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De Novo Synthesis of Dihydrobenzofurans and Indolines and Its Application to a Modular, Asymmetric Synthesis of Beraprost

[Image: see text] Dihydrobenzofurans and indolines are important constituents of pharmaceuticals. Herein, we describe a novel strategy for their construction in which the aromatic ring is created de novo through an inverse-electron demand Diels–Alder reaction and cheletropic extrusion sequence of a...

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Detalles Bibliográficos
Autores principales:	Wang, Ze-Shu, Bennett, Steven H., Kicin, Bilal, Jing, Changcheng, Pradeilles, Johan A., Thai, Karen, Smith, James R., Bacoş, P. David, Fasano, Valerio, Saunders, Carla M., Aggarwal, Varinder K.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2023
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10311537/ https://www.ncbi.nlm.nih.gov/pubmed/37326516 http://dx.doi.org/10.1021/jacs.3c04582

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