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Discovery of indolizine lactones as anticancer agents and their optimization through late-stage functionalization
Indolizines fused with a seven-member lactone ring were identified as a promising scaffold in the search for new anticancer agents. Through a modular synthetic sequence, a library of cis and trans indolizines lactones had their antiproliferative activity evaluated against hormone-refractory prostate...
Autores principales: | da Silva, Thiago Sabino, da Silva Souza, Matheus, Andricopulo, Adriano Defini, Coelho, Fernando |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
The Royal Society of Chemistry
2023
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10321224/ https://www.ncbi.nlm.nih.gov/pubmed/37416908 http://dx.doi.org/10.1039/d3ra03395c |
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