Cargando…
Structural Optimization of BIPPO Analogs as Potent Antimalarials
Malaria continues to pose a significant health threat, causing thousands of deaths each year. The limited availability of vaccines and medications, combined with the emergence of drug resistance, further complicates the fight against this disease. In this study, we aimed to enhance the antimalarial...
Autores principales: | Zheng, Yang, Matheeussen, An, Maes, Louis, Caljon, Guy, Sterk, Geert Jan, Leurs, Rob |
---|---|
Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
MDPI
2023
|
Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10343887/ https://www.ncbi.nlm.nih.gov/pubmed/37446602 http://dx.doi.org/10.3390/molecules28134939 |
Ejemplares similares
-
Discovery of
5-Phenylpyrazolopyrimidinone Analogs
as Potent Antitrypanosomal Agents with In Vivo Efficacy
por: Zheng, Yang, et al.
Publicado: (2023) -
Structure‐Activity Relationship of Phenylpyrazolones against Trypanosoma cruzi
por: Sijm, Maarten, et al.
Publicado: (2020) -
Structure Activity Relationship of N-Substituted Phenyldihydropyrazolones Against Trypanosoma cruzi Amastigotes
por: Sijm, Maarten, et al.
Publicado: (2021) -
3-nitroimidazo[1,2-b]pyridazine as a novel scaffold for antiparasitics with sub-nanomolar anti-Giardia lamblia activity
por: Zheng, Yang, et al.
Publicado: (2022) -
Chloroquine analogs as antimalarial candidates with potent in vitro and in vivo activity
por: Aguiar, Anna C.C., et al.
Publicado: (2018)