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Development of an Affinity-Based Probe to Profile Endogenous Human Adenosine A(3) Receptor Expression
[Image: see text] The adenosine A(3) receptor (A(3)AR) is a G protein-coupled receptor (GPCR) that exerts immunomodulatory effects in pathophysiological conditions such as inflammation and cancer. Thus far, studies toward the downstream effects of A(3)AR activation have yielded contradictory results...
Autores principales: | Beerkens, Bert L. H., Snijders, Inge M., Snoeck, Joep, Liu, Rongfang, Tool, Anton T. J., Le Dévédec, Sylvia E., Jespers, Willem, Kuijpers, Taco W., van Westen, Gerard J.P., Heitman, Laura H., IJzerman, Adriaan P., van der Es, Daan |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
American Chemical Society
2023
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Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10461224/ https://www.ncbi.nlm.nih.gov/pubmed/37531576 http://dx.doi.org/10.1021/acs.jmedchem.3c00854 |
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