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7-[(18)F]Fluoro-8-azaisatoic Anhydrides: Versatile Prosthetic Groups for the Preparation of PET Tracers

[Image: see text] (18)F-Fluorination of sensitive molecules is often challenging, but can be accomplished under suitably mild conditions using radiofluorinated prosthetic groups (PGs). Herein, 1-alkylamino-7-[(18)F]fluoro-8-azaisatoic anhydrides ([(18)F]AFAs) are introduced as versatile (18)F-labele...

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Detalles Bibliográficos
Autores principales:	Gröner, Benedikt, Willmann, Michael, Donnerstag, Lisa, Urusova, Elizaveta A., Neumaier, Felix, Humpert, Swen, Endepols, Heike, Neumaier, Bernd, Zlatopolskiy, Boris D.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2023
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10510393/ https://www.ncbi.nlm.nih.gov/pubmed/37625106 http://dx.doi.org/10.1021/acs.jmedchem.3c01310

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