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Data sets of human and mouse protein kinase inhibitors with curated activity data including covalent inhibitors
AIM: Generation of high-quality data sets of protein kinase inhibitors (PKIs). METHODOLOGY: Publicly available PKIs with reliable activity data were curated. PKIs with very weak activity were classified as inactive. Analogue series and PKIs containing reactive groups (warheads) enabling covalent inh...
Autores principales: | Xerxa, Elena, Bajorath, Jürgen |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Future Science Ltd
2023
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10518807/ https://www.ncbi.nlm.nih.gov/pubmed/37752915 http://dx.doi.org/10.2144/fsoa-2023-0088 |
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