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Side-Chain Modified [(99m)Tc]Tc-DT1 Mimics: A Comparative Study in NTS(1)R-Positive Models

Radiolabeled neurotensin analogs have been developed as candidates for theranostic use against neurotensin subtype 1 receptor (NTS(1)R)-expressing cancer. However, their fast degradation by two major peptidases, neprilysin (NEP) and angiotensin-converting enzyme (ACE), has hitherto limited clinical...

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Detalles Bibliográficos
Autores principales:	Kanellopoulos, Panagiotis, Nock, Berthold A., Rouchota, Maritina, Loudos, George, Krenning, Eric P., Maina, Theodosia
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	MDPI 2023
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10647616/ https://www.ncbi.nlm.nih.gov/pubmed/37958525 http://dx.doi.org/10.3390/ijms242115541

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