Cargando…

Novel Scaffolds Based on Bis-thiazole Connected to Quinoxaline or Thienothiophene through 2-Phenoxy-N-arylacetamide Groups as New Hybrid Molecules: Synthesis, Antibacterial Activity, and Molecular Docking Investigations

[Image: see text] The resistance of microorganisms to antimicrobials has endangered the health of many people across the world. Overcoming the resistance problem will require the invention of molecules with a new mechanism of action so that no cross-resistance with existing therapies occurs. Because...

Descripción completa

Detalles Bibliográficos
Autores principales:	Salem, Mostafa E., Abdullah, Abbas H., Ibrahim, Nada S., Zaki, Magdi E. A., Elwahy, Ahmed H. M., Abdelhamid, Ismail A.
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	American Chemical Society 2023
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC10666262/ https://www.ncbi.nlm.nih.gov/pubmed/38027350 http://dx.doi.org/10.1021/acsomega.3c07125

Ejemplares similares

An efficient synthesis of 4-phenoxy-quinazoline, 2-phenoxy-quinoxaline, and 2-phenoxy-pyridine derivatives using aryne chemistry
por: Zilla, Mahesh K., et al.
Publicado: (2021)

Reactions of Some New Thienothiophene Derivatives
por: Mabkhot, Yahia Nasser, et al.
Publicado: (2011)

Identification of Cyclic Sulfonamides with an N-Arylacetamide Group as α-Glucosidase and α-Amylase Inhibitors: Biological Evaluation and Molecular Modeling
por: Saddique, Furqan Ahmad, et al.
Publicado: (2022)

Isolation and characterization of arylacetamide deacetylase in cynomolgus macaques
por: UNO, Yasuhiro, et al.
Publicado: (2015)

Arylacetamide Deacetylase Is Involved in Vicagrel Bioactivation in Humans
por: Jiang, Jinfang, et al.
Publicado: (2017)

Design, Synthesis, Anticancer Activity and Molecular Docking of New 1,2,3-Triazole-Based Glycosides Bearing 1,3,4-Thiadiazolyl, Indolyl and Arylacetamide Scaffolds
por: Elganzory, Hussein H., et al.
Publicado: (2022)

(S)-Ethyl 2-[4-(6-chloroquinoxalin-2-yloxy)phenoxy]propanoate
por: Hu, Jun, et al.
Publicado: (2009)

Synthesis and Chemical Characterisation of Some New Diheteroaryl Thienothiophene Derivatives
por: Mabkhot, Yahia Nasser, et al.
Publicado: (2011)

Tin(ii) chloride dihydrate/choline chloride deep eutectic solvent: redox properties in the fast synthesis of N-arylacetamides and indolo(pyrrolo)[1,2-a]quinoxalines
por: Trujillo, Sergio Alfonso, et al.
Publicado: (2020)

Substitutions of Fluorine Atoms and Phenoxy Groups in the Synthesis of Quinoxaline 1,4-di-N-oxide Derivatives†
por: Vicente, Esther, et al.
Publicado: (2008)

Selective adsorptive separation of cyclohexane over benzene using thienothiophene cages
por: Ding, Yanjun, et al.
Publicado: (2021)

Synthesis, Molecular Docking, and Dynamic Simulation Targeting Main Protease (Mpro) of New, Thiazole Clubbed Pyridine Scaffolds as Potential COVID-19 Inhibitors
por: Alghamdi, Adel, et al.
Publicado: (2023)

A facile synthesis, and antimicrobial and anticancer activities of some pyridines, thioamides, thiazole, urea, quinazoline, β-naphthyl carbamate, and pyrano[2,3-d]thiazole derivatives
por: Zaki, Yasser H., et al.
Publicado: (2018)

Synthesis, Molecular Docking Study, and Cytotoxic Activity against MCF Cells of New Thiazole–Thiophene Scaffolds
por: Gomha, Sobhi M., et al.
Publicado: (2022)

Novel Bis-Thiazole Derivatives: Synthesis and Potential Cytotoxic Activity Through Apoptosis With Molecular Docking Approaches
por: Dawood, Kamal M., et al.
Publicado: (2021)

Characterization, comparative, and functional analysis of arylacetamide deacetylase from Gnathostomata organisms
por: Diaz-Vidal, Tania, et al.
Publicado: (2022)

An effective uranium removal using diversified synthesized cross-linked chitosan bis-aldehyde Schiff base derivatives from aqueous solutions
por: Hamed, Amira, et al.
Publicado: (2022)

Synthesis of novel antibacterial and antifungal quinoxaline derivatives
por: Tang, Xuemei, et al.
Publicado: (2022)

Signature of arylacetamide deacetylase expression is associated with prognosis and immune infiltration in ovarian cancer
por: Feng, Jianyang, et al.
Publicado: (2022)

Copper-catalyzed transformation of alkyl nitriles to N-arylacetamide using diaryliodonium salts
por: Sallio, Romain, et al.
Publicado: (2021)

[3.3]Dithia-bridged cyclophanes featuring a thienothiophene ring: synthesis, structures and conformational analysis
por: Mashraqui, Sabir H, et al.
Publicado: (2009)

Fluorescent Thienothiophene-Containing Squaraine Dyes and Threaded Supramolecular Complexes with Tunable Wavelengths between 600–800 nm
por: Liu, Wenqi, et al.
Publicado: (2018)

New Conjugates of Quinoxaline as Potent Antitubercular and Antibacterial Agents
por: Peraman, Ramalingam, et al.
Publicado: (2016)

Tetra-μ-benzoato-bis[(quinoxaline)copper(II)]
por: Lee, Eun Yong, et al.
Publicado: (2008)

Design, Synthesis and Anticancer Activity of New Polycyclic: Imidazole, Thiazine, Oxathiine, Pyrrolo-Quinoxaline and Thienotriazolopyrimidine Derivatives
por: Abu-Hashem, Ameen Ali, et al.
Publicado: (2021)

Thiazole Ring—A Biologically Active Scaffold
por: Petrou, Anthi, et al.
Publicado: (2021)

Synthesis of novel star-shaped molecules based on a 1,3,5-triazine core linked to different heterocyclic systems as novel hybrid molecules
por: Diab, Hadeer M., et al.
Publicado: (2020)

Thiazole-Based Thiosemicarbazones: Synthesis, Cytotoxicity Evaluation and Molecular Docking Study
por: Gomha, Sobhi M, et al.
Publicado: (2021)

Design of Thienothiophene-Based Copolymers with Various Side Chain-End Groups for Efficient Polymer Solar Cells
por: Chao, Ying-Chieh, et al.
Publicado: (2020)

Quinoxaline Moiety: A Potential Scaffold against Mycobacterium tuberculosis
por: Montana, Marc, et al.
Publicado: (2021)

2,3-Bis(4-ethoxyphenyl)quinoxaline
por: Ye, Ping-Ping, et al.
Publicado: (2009)

2,3-Bis(4-bromophenyl)quinoxaline
por: Jian, Fang-Fang, et al.
Publicado: (2007)

2,3-Bis(thiophen-3-yl)quinoxaline
por: Crundwell, Guy, et al.
Publicado: (2013)

2,3-Bis(phenoxymethyl)buta-1,3-diene
por: Sathiyanarayanan, K., et al.
Publicado: (2007)

Synthesis and biological evaluation of new derivatives of thieno-thiazole and dihydrothiazolo-thiazole scaffolds integrated with a pyrazoline nucleus as anticancer and multi-targeting kinase inhibitors
por: Othman, Ismail M. M., et al.
Publicado: (2021)

Design and synthesis of new bis(1,2,4-triazolo[3,4-b][1,3,4]thiadiazines) and bis((quinoxalin-2-yl)phenoxy)alkanes as anti-breast cancer agents through dual PARP-1 and EGFR targets inhibition
por: Thabet, Fatma M., et al.
Publicado: (2022)

1,4-Bis{4-[bis(prop-2-yn-1-yl)amino]phenoxy}benzene
por: Shah, Kiramat, et al.
Publicado: (2011)

Synthesis and α-Glucosidase Inhibition Activity of 2-[3-(Benzoyl/4-bromobenzoyl)-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl]-N-arylacetamides: An In Silico and Biochemical Approach
por: Saddique, Furqan Ahmad, et al.
Publicado: (2021)

Synthesis of Thymidine Phosphorylase Inhibitor Based on Quinoxaline Derivatives and Their Molecular Docking Study
por: Almandil, Noor Barak, et al.
Publicado: (2019)

1,4-Bis[2-(prop-1-enyl)phenoxy]butane
por: Bayramov, Musa R., et al.
Publicado: (2011)

Cannot write session to /tmp/vufind_sessions/sess_a0pv8qjd6c3j2a9oq0rl8g0eha