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Pyrazolo-triazolo-pyrimidines as adenosine receptor antagonists: A complete structure–activity profile
In the last 5 years, many efforts have been conducted searching potent and selective human A(3) adenosine antagonists. In this field several different classes of compounds, possessing very good affinity (nM range) and with a broad range of selectivity, have been proposed. Recently, our group synthes...
Autores principales: | Cacciari, Barbara, Bolcato, Chiara, Spalluto, Giampiero, Klotz, Karl-Norbet, Bacilieri, Magdalena, Deflorian, Francesca, Moro, Stefano |
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Formato: | Texto |
Lenguaje: | English |
Publicado: |
Kluwer Academic Publishers
2006
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC2096643/ https://www.ncbi.nlm.nih.gov/pubmed/18404432 http://dx.doi.org/10.1007/s11302-006-9027-x |
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