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Dequalinium: A Novel, High-affinity Blocker of CNGA1 Channels

Cyclic nucleotide–gated (CNG) channels have been shown to be blocked by diltiazem, tetracaine, polyamines, toxins, divalent cations, and other compounds. Dequalinium is an organic divalent cation which suppresses the rat small conductance Ca(2+)-activated K(+) channel 2 (rSK2) and the activity of pr...

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Detalles Bibliográficos
Autores principales:	Rosenbaum, Tamara, Islas, León D., Carlson, Anne E., Gordon, Sharona E.
Formato:	Texto
Lenguaje:	English
Publicado:	The Rockefeller University Press 2003
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC2217319/ https://www.ncbi.nlm.nih.gov/pubmed/12508052 http://dx.doi.org/10.1085/jgp.20028716

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