Cargando…

Receptor-Drug Interaction: Europium Employment for Studying the Biochemical Pathway of G-Protein-Coupled Receptor Activation

In medicinal chemistry field, the biochemical pathways, involved in 7-transmembrane domains G-protein coupled receptors (GPCRs) activation, are commonly studied to establish the activity of ligands towards GPCRs. The most studied steps are the measurement of activated GTP-α subunit and stimulated in...

Descripción completa

Detalles Bibliográficos
Autores principales:	Antonio, Colabufo Nicola, Grazia, Perrone Maria, Marialessandra, Contino, Francesco, Berardi, Roberto, Perrone
Formato:	Texto
Lenguaje:	English
Publicado:	Hindawi Publishing Corporation 2007
Materias:	Review Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC2266097/ https://www.ncbi.nlm.nih.gov/pubmed/18350113 http://dx.doi.org/10.1155/2007/12635

Ejemplares similares

Why PB28 Could Be a Covid 2019 Game Changer?
por: Colabufo, Nicola Antonio, et al.
Publicado: (2020)

PB28, the Sigma-1 and Sigma-2 Receptors Modulator With Potent Anti–SARS-CoV-2 Activity: A Review About Its Pharmacological Properties and Structure Affinity Relationships
por: Abate, Carmen, et al.
Publicado: (2020)

An innovative small molecule for promoting neuroreparative strategies
por: Colabufo, Nicola Antonio, et al.
Publicado: (2018)

Overcoming Multidrug Resistance (MDR): Design, Biological Evaluation and Molecular Modelling Studies of 2,4‐Substituted Quinazoline Derivatives
por: Braconi, Laura, et al.
Publicado: (2022)

Editorial: The CB2 Cannabinoid System: A New Strategy in Neurodegenerative Disorder and Neuroinflammation
por: Contino, Marialessandra, et al.
Publicado: (2017)

6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers
por: Braconi, Laura, et al.
Publicado: (2020)

The interaction of celecoxib with MDR transporters enhances the activity of mitomycin C in a bladder cancer cell line
por: Pagliarulo, Vincenzo, et al.
Publicado: (2013)

Small and Innovative Molecules as New Strategy to Revert MDR
por: Zinzi, Laura, et al.
Publicado: (2014)

ABC transporters in CSCs membranes as a novel target for treating tumor relapse
por: Zinzi, Laura, et al.
Publicado: (2014)

Inhibition of hERG potassium channel by the antiarrhythmic agent mexiletine and its metabolite m-hydroxymexiletine
por: Gualdani, Roberta, et al.
Publicado: (2015)

miRNAs for the Detection of MultiDrug Resistance: Overview and Perspectives
por: Gisel, Andreas, et al.
Publicado: (2014)

Small-animal PET evaluation of [(11)C]MC113 as a PET tracer for P-glycoprotein
por: Mairinger, Severin, et al.
Publicado: (2010)

Multi-Target Directed Ligands (MTDLs) Binding the σ(1) Receptor as Promising Therapeutics: State of the Art and Perspectives
por: Abatematteo, Francesca Serena, et al.
Publicado: (2021)

New Strategies to Overcome Resistance to Chemotherapy and Immune System in Cancer
por: Riganti, Chiara, et al.
Publicado: (2019)

Selective κ Opioid Antagonists nor-BNI, GNTI and JDTic Have Low Affinities for Non-Opioid Receptors and Transporters
por: Munro, Thomas A., et al.
Publicado: (2013)

Receptor–Receptor Interactions of G Protein-Coupled Receptors in the Carotid Body: A Working Hypothesis
por: Porzionato, Andrea, et al.
Publicado: (2018)

Editorial: The Canonical and Non-Canonical Endocannabinoid System as a Target in Cancer and Acute and Chronic Pain
por: Contino, Marialessandra, et al.
Publicado: (2020)

Editorial: Molecular modulators of GPCRs signal transduction
por: Vrecl, Milka, et al.
Publicado: (2023)

Structural Characterization of Receptor–Receptor Interactions in the Allosteric Modulation of G Protein-Coupled Receptor (GPCR) Dimers
por: Lazim, Raudah, et al.
Publicado: (2021)

Receptor–Receptor Interactions and Glial Cell Functions with a Special Focus on G Protein-Coupled Receptors
por: Guidolin, Diego, et al.
Publicado: (2021)

PRECOG: PREdicting COupling probabilities of G-protein coupled receptors
por: Singh, Gurdeep, et al.
Publicado: (2019)

Effects of Europium Complex on Thermal and Photoluminescence Properties of Polyurethane-Europium Materials
por: Gao, Lijun, et al.
Publicado: (2023)

G protein-coupled receptors /
Publicado: (2000)

G-Protein-Coupled Receptors
por: Thiriet, Marc
Publicado: (2011)

Evolution of a G protein-coupled receptor response by mutations in regulatory network interactions
por: Di Roberto, Raphaël B., et al.
Publicado: (2016)

Structural Insights into Ligand—Receptor Interactions Involved in Biased Agonism of G-Protein Coupled Receptors
por: Jóźwiak, Krzysztof, et al.
Publicado: (2021)

Evidence for Protein–Protein Interaction between Dopamine Receptors and the G Protein-Coupled Receptor 143
por: Bueschbell, Beatriz, et al.
Publicado: (2021)

Unraveling the Functional Significance of Unstructured Regions in G Protein-Coupled Receptors
por: Maggio, Roberto, et al.
Publicado: (2023)

G protein–receptor kinases 5/6 are the key regulators of G protein–coupled receptor 35–arrestin interactions
por: Ganguly, Amlan, et al.
Publicado: (2023)

Mapping Interactions of Microbial Metabolites with Human G-Protein-Coupled Receptors
por: Colosimo, Dominic A., et al.
Publicado: (2019)

Integration and Spatial Organization of Signaling by G Protein-Coupled Receptor Homo- and Heterodimers
por: Maggio, Roberto, et al.
Publicado: (2021)

Fluorescence based HTS-compatible ligand binding assays for dopamine D(3) receptors in baculovirus preparations and live cells
por: Tahk, Maris-Johanna, et al.
Publicado: (2023)

G Protein-Coupled Receptors in Cancer
por: Bar-Shavit, Rachel, et al.
Publicado: (2016)

G-protein-coupled Receptors in Fungi
por: El-Defrawy, Mohamed M. H., et al.
Publicado: (2020)

G Protein-Coupled Receptors in Osteoarthritis
por: Wang, Fanhua, et al.
Publicado: (2022)

A Rapid and Efficient Immunoenzymatic Assay to Detect Receptor Protein Interactions: G Protein-Coupled Receptors
por: Zappelli, Elisa, et al.
Publicado: (2014)

Functional Interaction of Endothelin Receptors in Mediating Natriuresis Evoked by G Protein–Coupled Estrogen Receptor 1
por: Gohar, Eman Y., et al.
Publicado: (2021)

The multiple combination of Paclitaxel, Ramucirumab and Elacridar reverses the paclitaxel-mediated resistance in gastric cancer cell lines
por: Schirizzi, Annalisa, et al.
Publicado: (2023)

Silver europium(III) polyphosphate
por: Ayadi, Mounir, et al.
Publicado: (2009)

G-Protein coupled receptors: structure and function in drug discovery
por: Odoemelam, Chiemela S., et al.
Publicado: (2020)

Cannot write session to /tmp/vufind_sessions/sess_gk4maarp7kq2l37001c0bj03d1