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Antagonist affinity measurements at the Gi-coupled human histamine H3 receptor expressed in CHO cells
BACKGROUND: The H3 histamine receptor is a Gi-coupled GPCR that has been proven to exist in different agonist-induced states, including that defined by the protean agonist proxyfan. Several GPCRs are now known to exist in different states. For some of these, antagonist affinity measurement remain co...
Autor principal: | Baker, Jillian G |
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Formato: | Texto |
Lenguaje: | English |
Publicado: |
BioMed Central
2008
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC2430196/ https://www.ncbi.nlm.nih.gov/pubmed/18538007 http://dx.doi.org/10.1186/1471-2210-8-9 |
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