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Allosteric Modulation of the Calcium-Sensing Receptor
The calcium (Ca(2+))-sensing receptor (CaR) belongs to family C of the G-protein coupled receptors (GPCRs). The receptor is activated by physiological levels of Ca(2+) (and Mg(2+)) and positively modulated by a range of proteinogenic L-α-amino acids. Recently, several synthetic allosteric modulators...
Autores principales: | Jensen, Anders A, Bräuner-Osborne, Hans |
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Formato: | Texto |
Lenguaje: | English |
Publicado: |
Bentham Science Publishers Ltd.
2007
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC2656812/ https://www.ncbi.nlm.nih.gov/pubmed/19305800 http://dx.doi.org/10.2174/157015907781695982 |
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