Cargando…

Synthesis of Novel 3-Aryl-N-Methyl-1,2,5,6-Tetrahydropyridine Derivatives by Suzuki coupling: As Acetyl Cholinesterase Inhibitors

Alzheimer’s disease (AD) is a neurodegenerative disorder affecting the central nervous system, which is also associated with progressive loss of memory and cognition. The development of numerous structural classes of compounds with different pharmacological profile could be an evolving, promising th...

Descripción completa

Detalles Bibliográficos
Autores principales:	Prasad, S.B. Benaka, Kumar, Y.C. Sunil, Kumar, C.S. Ananda, Sadashiva, C.T, Vinaya, K, Rangappa, K.S
Formato:	Texto
Lenguaje:	English
Publicado:	Bentham Science Publishers Ltd. 2007
Materias:	Article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC2709467/ https://www.ncbi.nlm.nih.gov/pubmed/19662135 http://dx.doi.org/10.2174/1874104500701010004

Ejemplares similares

1-Acetyl-2-r,6-c-bis(4-chlorophenyl)-3-methyl-1,2,5,6-tetrahydropyridin-4-yl acetate
por: Vimalraj, V., et al.
Publicado: (2010)

Ethyl 4-hydroxy-2,6-diphenyl-1-[2-(piperidin-1-yl)acetyl]-1,2,5,6-tetrahydropyridine-3-carboxylate
por: Aridoss, G., et al.
Publicado: (2010)

4-Ethynyl-2,2,6,6-tetramethyl-1,2,5,6-tetrahydropyridine N-oxide
por: Bats, Jan W., et al.
Publicado: (2009)

Methyl 2,6-diphenyl-1-p-tolyl-4-(p-tolylamino)-1,2,5,6-tetrahydropyridine-3-carboxylate
por: Venugopala, K. N., et al.
Publicado: (2012)

Ethyl 1-[2-(1H-benzotriazol-1-yl)acetyl]-4-hydroxy-2,6-diphenyl-1,2,5,6-tetrahydropyridine-3-carboxylate
por: Aridoss, G., et al.
Publicado: (2011)

Ethyl 1-benzoyl-4-hydroxy-2,6-diphenyl-1,2,5,6-tetrahydropyridine-3-carboxylate
por: Aridoss, G., et al.
Publicado: (2011)

Ethyl 1-[2-(1,3-benzoxazol-2-ylsulfanyl)acetyl]-4-hydroxy-2,6-diphenyl-1,2,5,6-tetrahydropyridine-3-carboxylate
por: Aridoss, G., et al.
Publicado: (2011)

Ethyl 4-anilino-2,6-bis(4-fluorophenyl)-1-phenyl-1,2,5,6-tetrahydropyridine-3-carboxylate
por: Anthal, Sumati, et al.
Publicado: (2013)

Cobalt‐Catalyzed Suzuki Biaryl Coupling of Aryl Halides
por: Asghar, Soneela, et al.
Publicado: (2017)

Single crystal X-ray structural and Hirshfeld surface analysis dataset for some isobutyl-1,2,6-triaryl-4-(arylamino)-1,2,5,6-tetrahydropyridine-3-carboxylates
por: Kumar, Chandran Udhaya, et al.
Publicado: (2021)

Ethyl 4-hydroxy-2,6-diphenyl-1-(2-thiomorpholinoacetyl)-1,2,5,6-tetrahydropyridine-3-carboxylate
por: Aridoss, G., et al.
Publicado: (2010)

Ethyl 1-(2-bromopropanoyl)-4-hydroxy-2,6-diphenyl-1,2,5,6-tetrahydropyridine-3-carboxylate
por: Aridoss, G., et al.
Publicado: (2009)

DNA-Compatible Suzuki-Miyaura Cross-Coupling Reaction of Aryl Iodides With (Hetero)Aryl Boronic Acids for DNA-Encoded Libraries
por: Siripuram, Vijay Kumar, et al.
Publicado: (2022)

Methyl 4-(4-fluoroanilino)-1,2,6-tris(4-fluorophenyl)-1,2,5,6-tetrahydropyridine-3-carboxylate
por: Anthal, Sumati, et al.
Publicado: (2013)

Ethyl 4-hydroxy-1-(2-morpholinopropanoyl)-2,6-diphenyl-1,2,5,6-tetrahydropyridin-3-carboxylate
por: Aridoss, G., et al.
Publicado: (2009)

Ethyl 4-hydroxy-2,6-diphenyl-1-(2-thiomorpholinopropanoyl)-1,2,5,6-tetrahydropyridine-3-carboxylate
por: Aridoss, G., et al.
Publicado: (2009)

(R)-(+)-Dimethyl[4-oxido-2-oxo-1-(1-phenylethyl)-1,2,5,6-tetrahydropyridin-3-yl]sulfonium
por: Gordillo, Paola G., et al.
Publicado: (2011)

Ethyl 4-anilino-2,6-bis(4-chlorophenyl)-1-phenyl-1,2,5,6-tetrahydropyridine-3-carboxylate
por: Yu, Jianfeng, et al.
Publicado: (2013)

Screening and analysis of acetyl-cholinesterase (AChE) inhibitors in the context of Alzheimer's disease
por: Khan, Mohd. Babu, et al.
Publicado: (2018)

Memantine combined with an acetyl cholinesterase inhibitor – hope for the future?
por: Fox, Chris, et al.
Publicado: (2006)

Neuroprotective derivatives of tacrine that target NMDA receptor and acetyl cholinesterase – Design, synthesis and biological evaluation
por: Remya, Chandran, et al.
Publicado: (2021)

Ethyl 2,6-bis(4-chlorophenyl)-4-(4-fluoroanilino)-1-(4-fluorophenyl)-1,2,5,6-tetrahydropyridine-3-carboxylate
por: Anthal, Sumati, et al.
Publicado: (2013)

Ethyl 2,6-bis(4-chlorophenyl)-4-(4-methylanilino)-1-(4-methylphenyl)-1,2,5,6-tetrahydropyridine-3-carboxylate
por: Anthal, Sumati, et al.
Publicado: (2013)

Suzuki-Miyaura Coupling Enabled by Aryl to Vinyl 1,4-Palladium Migration
por: Li, Meng-Yao, et al.
Publicado: (2020)

Asymmetric Suzuki-Miyaura coupling of heterocycles via Rhodium-catalysed allylic arylation of racemates
por: Schäfer, Philipp, et al.
Publicado: (2017)

A direct method to visualise the aryl acylamidase activity on cholinesterases in polyacrylamide gels
por: Jaganathan, Lakshmanan, et al.
Publicado: (2000)

Serum Acetyl Cholinesterase as a Biomarker of Arsenic Induced Neurotoxicity in Sprague-Dawley Rats
por: Patlolla, Anita K., et al.
Publicado: (2005)

Acetyl and butyryl cholinesterase inhibitory sesquiterpene lactones from Amberboa ramosa
por: Ibrahim, Muhammad, et al.
Publicado: (2013)

Crystal structure of 1′-(2-methylpropyl)-2,3-dihydrospiro[1-benzothiopyran-4,4′-imidazolidine]-2′,5′-dione
por: Theodore, Cynthia E., et al.
Publicado: (2014)

Synthesis, spectroscopic, topological, hirshfeld surface analysis, and anti-covid-19 molecular docking investigation of isopropyl 1-benzoyl-4-(benzoyloxy)-2,6-diphenyl-1,2,5,6-tetrahydropyridine-3-carboxylate
por: Ramalingam, Arulraj, et al.
Publicado: (2022)

Carbonylative Suzuki Couplings of Aryl Bromides with Boronic Acid Derivatives under Base-Free Conditions
por: Bjerglund, Klaus M., et al.
Publicado: (2014)

An Efficient Synthesis of Aryl-Substituted Pyrroles by the Suzuki–Miyaura Coupling Reaction of SEM-Protected Pyrroles
por: Cui, Keli, et al.
Publicado: (2019)

Synthesis and Functionalization of Challenging meso-Substituted Aryl Bis-pocket Porphyrins Accessed via Suzuki–Miyaura Cross-Coupling
por: Droege, Daniel G., et al.
Publicado: (2022)

Author Correction: Asymmetric Suzuki-Miyaura coupling of heterocycles via Rhodium-catalysed allylic arylation of racemates
por: Schäfer, Philipp, et al.
Publicado: (2018)

An expedient, mild and aqueous method for Suzuki–Miyaura diversification of (hetero)aryl halides or (poly)chlorinated pharmaceuticals
por: Sharma, Sunil V., et al.
Publicado: (2021)

Synthesis, crystal structure, Hirshfeld surface analysis, DFT and NBO study of ethyl 1-(4-fluorophenyl)-4-[(4-fluorophenyl)amino]-2,6-diphenyl-1,2,5,6-tetrahydropyridine-3-carboxylate
por: Bansal, Ravi, et al.
Publicado: (2023)

Crystal structure of poly[μ(2)-aqua-aqua(μ(2)-4-nitro-2,5,6-trioxo-1,2,5,6-tetrahydropyridin-3-olato)hemi-μ(4)-oxalato-barium(II)]
por: Alabada, Rusul, et al.
Publicado: (2015)

DNA‐Encoded Libraries: Aryl Fluorosulfonates as Versatile Electrophiles Enabling Facile On‐DNA Suzuki, Sonogashira, and Buchwald Reactions
por: Xu, Hongtao, et al.
Publicado: (2019)

New biomaterials for Ni biosorption turned into catalysts for Suzuki–Miyaura cross coupling of aryl iodides in green conditions
por: Cases, Lucie, et al.
Publicado: (2021)

1256. Antiretroviral Switching in Colombia: A Retrospective Cohort Study.
por: Forero, Shirley Vanessa Correa, et al.
Publicado: (2022)

Cannot write session to /tmp/vufind_sessions/sess_018hgtcskpubjk75kalnjt6d30