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Sleep-promoting action of IIK7, a selective MT(2) melatonin receptor agonist in the rat
Several novel melatonin receptor agonists, in addition to various formulations of melatonin itself, are either available or in development for the treatment of insomnia. Melatonin is thought to exert its effects principally through two high affinity, G-protein coupled receptors, MT(1) and MT(2), tho...
Autores principales: | Fisher, Simon P., Sugden, David |
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Formato: | Texto |
Lenguaje: | English |
Publicado: |
Elsevier Scientific Publishers Ireland
2009
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC2724036/ https://www.ncbi.nlm.nih.gov/pubmed/19429170 http://dx.doi.org/10.1016/j.neulet.2009.04.005 |
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