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Differential regulation of muscarinic M(1 )receptors by orthosteric and allosteric ligands

BACKGROUND: Activation of muscarinic M(1 )receptors is mediated via interaction of orthosteric agonists with the acetylcholine binding site or via interaction of allosteric agonists with different site(s) on the receptor. The focus of the present study was to determine if M(1 )receptors activated by...

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Detalles Bibliográficos
Autores principales:	Davis, Christopher N, Bradley, Stefania Risso, Schiffer, Hans H, Friberg, Mikael, Koch, Kristian, Tolf, Bo-Ragnar, Bonhaus, Douglas W, Lameh, Jelveh
Formato:	Texto
Lenguaje:	English
Publicado:	BioMed Central 2009
Materias:	Research article
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC2794843/ https://www.ncbi.nlm.nih.gov/pubmed/19951444 http://dx.doi.org/10.1186/1471-2210-9-14

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