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Targeting ketone drugs towards transport by the intestinal peptide transporter, PepT1
Thiodipeptide prodrugs of the ketone nabumetone are shown to have affinity for, and be transported by, PepT1 in vitro.
Autores principales: | Foley, David, Bailey, Patrick, Pieri, Myrtani, Meredith, David |
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Formato: | Texto |
Lenguaje: | English |
Publicado: |
Royal Society of Chemistry
2009
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC2898646/ https://www.ncbi.nlm.nih.gov/pubmed/19262922 http://dx.doi.org/10.1039/b818606e |
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