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A Pharmacological Primer of Biased Agonism
Biased agonism is one of the fastest growing topics in G protein-coupled receptor pharmacology; moreover, biased agonists are used in the clinic today: carvedilol (Coreg(®)) is a biased agonist of beta-adrenergic receptors. However, there is a general lack of understanding of biased agonism when com...
Autor principal: | Andresen, Bradley T |
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Formato: | Online Artículo Texto |
Lenguaje: | English |
Publicado: |
Bentham Science Publishers Ltd
2011
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Materias: | |
Acceso en línea: | https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3182416/ https://www.ncbi.nlm.nih.gov/pubmed/21476970 http://dx.doi.org/10.2174/187153011795564179 |
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