Cargando…

Antiepileptic activity and subtype-selective action of flupirtine at GABA(A) receptors

Detalles Bibliográficos
Autores principales:	Bajrić, Mirnes, Klinger, Felicia, Schandl, Ulla, Kubista, Helmut, Boehm, Stefan
Formato:	Online Artículo Texto
Lenguaje:	English
Publicado:	BioMed Central 2012
Materias:	Meeting Abstract
Acceso en línea:	https://www.ncbi.nlm.nih.gov/pmc/articles/PMC3506359/ http://dx.doi.org/10.1186/2050-6511-13-S1-A90

Ejemplares similares

δ Subunit‐containing GABA(A) receptors are preferred targets for the centrally acting analgesic flupirtine
por: Klinger, Felicia, et al.
Publicado: (2015)

The non-opioid analgesic flupirtine is a modulator of GABA(A )receptors involved in pain sensation
por: Popovici, Felicia, et al.
Publicado: (2008)

The anticonvulsant retigabine is a subtype selective modulator of GABA (A) receptors
por: Treven, Marco, et al.
Publicado: (2015)

Understanding subtype-selective allosteric modulation of GABA(A) receptors
por: Puthenkalam, Roshan, et al.
Publicado: (2012)

Heterogeneity of release-regulating muscarinic receptors in rat sympathetic neurons: evidence for inhibitory presynaptic M(1 )receptors
por: Kubista, Helmut, et al.
Publicado: (2008)

The interplay of excitatory and inhibitory coupling modes is crucial for the regulation of neuronal electrical activities by L-type calcium channels
por: Geier, Petra, et al.
Publicado: (2010)

L-type voltage-gated calcium channels in hippocampal neurons and their potential as anti-epilept(ogen)ic drug targets
por: Geier, Petra, et al.
Publicado: (2009)

Current-clamp experiments on primary hippocampal neurons shed light on the role of L-type voltage-gated calcium channels in depolarization shifts
por: Kubista, Helmut, et al.
Publicado: (2011)

Functional implications of K(V)7 channel phosphorylation
por: Salzer, Isabella, et al.
Publicado: (2012)

Flupirtine: Clinical pharmacology
por: Harish, S, et al.
Publicado: (2012)

Raised Activity of L-Type Calcium Channels Renders Neurons Prone to Form Paroxysmal Depolarization Shifts
por: Rubi, Lena, et al.
Publicado: (2013)

Benzodiazepines modulate GABA(A )receptors by reducing a gamma-subunit-mediated inhibition of GABA sensitivity
por: Baburin, Igor, et al.
Publicado: (2009)

Facilitation of transmitter release from rat sympathetic neurons via presynaptic P2Y(1 )receptors
por: Chandaka, Giri K, et al.
Publicado: (2008)

EHMTI-0065. Effects of antiepileptic drugs on spreading depression in the chick retina: implications for migraine prophylaxis
por: Mascarenhas de Moraes, J, et al.
Publicado: (2014)

P2Y(1 )receptors are linked to K(Ca)2 channels in PC12 cells
por: Schicker, Klaus, et al.
Publicado: (2009)

Functional characterization of the antiepileptic drug candidate, padsevonil, on GABA(A) receptors
por: Niespodziany, Isabelle, et al.
Publicado: (2020)

Nucleotides excite sensory neurons via two P2Y receptors and a dual signaling cascade
por: Yousuf, Arsalan, et al.
Publicado: (2009)

Pharmacological Effect of GABA Analogues on GABA-ρ2 Receptors and Their Subtype Selectivity
por: Naffaa, Moawiah M., et al.
Publicado: (2022)

The GABA(A) receptor α2 subunit gene (GABRA2) is associated with alcohol-related behavior
por: Švob Štrac, Dubravka, et al.
Publicado: (2012)

Functional and physical interactions between P2Y receptors and ion channels
por: Gafar, Hend, et al.
Publicado: (2012)

Inhibition of Spontaneous Contractility of Isolated Caprine Ureter by Flupirtine
por: Naik, Girish S, et al.
Publicado: (2018)

Flupirtine derivatives as potential treatment for the neuronal ceroid lipofuscinoses
por: Makoukji, Joelle, et al.
Publicado: (2018)

Exogenous Flupirtine as Potential Treatment for CLN3 Disease
por: Maalouf, Katia, et al.
Publicado: (2020)

Flupirtine in the Management of Taxane-induced Pain in Cancer Patients
por: Paul, Anusha, et al.
Publicado: (2022)

Expression mRNA pattern of retinoic acid and retinoid X nuclear receptor subtypes in thyroid carcinomas
por: Brtko, Julius, et al.
Publicado: (2013)

Amphetamine actions rely on the availability of phosphatidylinositol-4,5-bisphosphate
por: Buchmayer, Florian, et al.
Publicado: (2011)

Absolute GABA spectroscopy with MEGA-PRESS and watermapping in sensorimotor and visual cortex and correlation to handedness
por: Oeltzschner, Georg, et al.
Publicado: (2014)

Antiepileptic Drugs and Their Dual Mechanism of Action on Carbonic Anhydrase
por: Magheru, Calin, et al.
Publicado: (2022)

Levetirazetam: antiepileptic-induced psychosis
por: Vilella Martín, C., et al.
Publicado: (2022)

Autoregulation in PC12 cells via P2Y receptors: Evidence for non-exocytotic nucleotide release from neuroendocrine cells
por: Hussl, Simon, et al.
Publicado: (2007)

GABA(A) receptor subtype selectivity of the proconvulsant rodenticide TETS
por: Pressly, Brandon, et al.
Publicado: (2017)

Novel Molecule Exhibiting Selective Affinity for GABA(A) Receptor Subtypes
por: Borghese, Cecilia M., et al.
Publicado: (2017)

A membrane network of receptors and enzymes for adenine nucleotides and nucleosides
por: Schicker, Klaus, et al.
Publicado: (2008)

Effect of flupirtine on the growth and viability of U373 malignant glioma cells
por: Panchanathan, Elango, et al.
Publicado: (2013)

Role of flupirtine as a preemptive analgesic in patients undergoing laparoscopic cholecystectomy
por: Yadav, Ghanshyam, et al.
Publicado: (2015)

Role of flupirtine in reducing preoperative anxiety of patients undergoing craniotomy procedure
por: Yadav, Ghanshyam, et al.
Publicado: (2017)

Efficacy of flupirtine for postoperative pain: A systematic review and meta-analysis
por: Dey, Samarjit, et al.
Publicado: (2023)

Discovery and biological evaluation of a diphenethylamine derivative (HS665), a highly potent and selective κ opioid receptor agonist
por: Spetea, Mariana, et al.
Publicado: (2012)

The Paroxysmal Depolarization Shift: Reconsidering Its Role in Epilepsy, Epileptogenesis and Beyond
por: Kubista, Helmut, et al.
Publicado: (2019)

Reclassifying ovarian cancer: origins, subtypes and resistance to therapy
por: Bowtell, DDL
Publicado: (2012)

Cannot write session to /tmp/vufind_sessions/sess_8jrq1kh8g2ugt5uqd4gislvptv